Search references for CB03 154. Phrases containing CB03 154
See searches and references containing CB03 154!CB03 154
Pharmaceutical compound
CB03-154 is a Kv7.2 and Kv7.3 potassium channel opener which is under development for the treatment of amyotrophic lateral sclerosis (ALS), epilepsy, major
CB03-154
Non-opioid analgesic drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Suzetrigine
Oral cough medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Benzonatate
Beta blocker drug
J, Court DS (eds.). Medical Sciences. Elsevier Health Sciences. pp. 101–154 [150]. ISBN 978-0-7020-5249-1. Young R, Glennon RA (April 2009). "S(-)Propranolol
Propranolol
Neurotoxin
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Tetrodotoxin
Medication against high blood pressure
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Amlodipine
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Meclizine
Medication used for epilepsy, bipolar disorder and migraine
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Valproate
Anticonvulsant medication
review from South Asia". Indian Journal of Psychological Medicine. 37 (2): 154–158. doi:10.4103/0253-7176.155613. PMC 4418246. PMID 25969599. Wang S, Zheng
Lamotrigine
Medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Etripamil
Experimental anticonvulsant
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Azetukalner
Drug for chronic pain
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Crisugabalin
Pharmaceutical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Relutrigine
Medication to treat high blood pressure and alopecia
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Minoxidil
Drug used to treat angina
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Ranolazine
Anti-seizure medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Phenytoin
Local anesthetic
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Lidocaine
Transmembrane protein allowing sodium ions in and out
(2000). Principles of Neural Science (4th ed.). New York: McGraw-Hill. pp. 154–69. ISBN 978-0-8385-7701-1.{{cite book}}: CS1 maint: multiple names: authors
Sodium_channel
Local anaesthetic drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Benzocaine
Sedating antidepressant
(3 and 6 mg) for the treatment of insomnia". Future Neurology. 6 (2): 143–154. doi:10.2217/fnl.10.83. ISSN 1479-6708. Dawkins K, Manji HK, Potter WZ (20
Doxepin
Local anesthetic drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Procaine
Anticonvulsant medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Oxcarbazepine
Muscle relaxant medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Baclofen
Benzodiazepine medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Lorazepam
Pharmaceutical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Flindokalner
Sterol biosynthesized by all animal cells
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Cholesterol
Antiarrhythmic medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Amiodarone
Class of medication used to treat high blood pressure
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Dihydropyridine calcium channel blockers
Dihydropyridine_calcium_channel_blockers
Opioid used to treat pain and opioid use disorder
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Buprenorphine
Family of transport proteins
extracellular immunoglobulin-like domain". The Journal of Cell Biology. 154 (2): 427–34. doi:10.1083/jcb.200102086. PMC 2150779. PMID 11470829. Antzelevitch
Voltage-gated_sodium_channel
Calcium channel blocker medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Diltiazem
Anticonvulsant medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Pregabalin
Muscle relaxant
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Chlorzoxazone
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Mirogabalin
Medication used to treat epilepsy and migraine
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Topiramate
Several medications which disrupt the movement of Na+ ions
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Sodium_channel_blocker
Antibiotic medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Erythromycin
Drugs that disrupt movement of calcium across calcium channels
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Calcium_channel_blocker
Medication used to treat ADHD
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Atomoxetine
Pharmaceutical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Naminidil
Gamma-aminobutyric acid analog
Cohort Study". Annals of Internal Medicine. 177 (Online ahead of print): 144–154. doi:10.7326/M23-0849. PMID 38224592. S2CID 266985259. Mersfelder TL, Nichols
Gabapentin
Antihistamine used to treat allergies
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Chlorphenamine
Antihypertensive drug of the calcium channel blocker class
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Nicardipine
Antiarrhythmic medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Flecainide
Peripheral D2 receptor antagonist
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Domperidone
Antihistamine medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Diphenhydramine
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Solifenacin
Pharmaceutical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Opakalim
Active metabolite of oxcarbazepine
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Licarbazepine
Calcium channel blocker medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Nifedipine
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Glipizide
Selective estrogen receptor modulator
Estrogen/antiestrogen Action and Breast Cancer Therapy. Univ of Wisconsin Press. pp. 28, 154. ISBN 978-0-299-10480-1. Pratt WB (1994). The Anticancer Drugs. Oxford University
Tamoxifen
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Roxithromycin
Antihypertensive drug of the calcium channel blocker class
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Barnidipine
Medication used to treat tuberculosis
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Bedaquiline
Antidepressant medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Nortriptyline
Class of depressant drugs derived from barbituric acid
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Barbiturate
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Terfenadine
Antihypertensive drug of the calcium channel blocker class
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Lercanidipine
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Cromakalim
Species of plant
Revision) Variation—Australia New Zealand Food Standards Code – Amendment No. 154 - 2015-gs1906 - New Zealand Gazette". gazette.govt.nz. Archived from the
Kava
Pore-forming membrane protein
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Ion_channel
Pair of enantiomers
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Mexiletine
Pharmaceutical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Fluoxakalner
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
PNU-282,987
Antibiotic medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Clarithromycin
Benzhydryl compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Tolterodine
Reversible monoamine oxidase B inhibitor
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Safinamide
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Piperocaine
Anticonvulsant medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Carbamazepine
Medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Sotalol
Pharmaceutical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Pynegabine
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Epithelial sodium channel blocker
Epithelial_sodium_channel_blocker
Index of articles associated with the same name
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Channel_opener
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Zonisamide
Skeletal muscle relaxant drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Tolperisone
Antihypertensive drug of the calcium channel blocker class
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Isradipine
Pain and blood pressure medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Amlodipine/celecoxib
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Nicorandil
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Mefenamic_acid
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Bencyclane
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Niguldipine
Antihypertensive drug of the calcium channel blocker class
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Nilvadipine
Paralytic shellfish toxin
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Saxitoxin
Mammalian protein found in humans
of the mammalian epididymis". Journal of Molecular Histology. 50 (2): 141–154. doi:10.1007/s10735-019-09813-3. PMID 30659401. S2CID 58026884. Sharma S
Cystic fibrosis transmembrane conductance regulator
Cystic_fibrosis_transmembrane_conductance_regulator
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Arbaclofen_placarbil
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Encainide
Medication
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Telmisartan/amlodipine/indapamide
Telmisartan/amlodipine/indapamide
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Bay_K8644
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
4-Methylpregabalin
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Pinacidil
Local anaesthetic drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Tetracaine
Drug for chronic pain
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Ziconotide
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Pheneturide
Antihistamine drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Astemizole
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Caroverine
List of pharmaceutical drugs under clinical development for treatment of depression
TS-1211; TS-121) – vasopressin V1b receptor antagonist CB-03 (CB-04; CB-003; CB03-154) – KCNQ2 and KCNQ3 potassium channel stimulant Centanafadine (CTN; EB-1020)
List of investigational antidepressants
List_of_investigational_antidepressants
Investigational analgesic drug
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
DSP-2230
Antifungal chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Ketoconazole
Chemical compound
(SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip
Gliclazide
travel, tourism, insurance
CB03 154
CB03 154
CB03 154
CB03 154
CB03 154
CB03 154
CB03 154
CB03 154
CB03 154
travel, tourism, insurance