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CB03 154

  • CB03-154
  • Pharmaceutical compound

    CB03-154 is a Kv7.2 and Kv7.3 potassium channel opener which is under development for the treatment of amyotrophic lateral sclerosis (ALS), epilepsy, major

    CB03-154

    CB03-154

    CB03-154

  • Suzetrigine
  • Non-opioid analgesic drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Suzetrigine

    Suzetrigine

    Suzetrigine

  • Benzonatate
  • Oral cough medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Benzonatate

    Benzonatate

  • Propranolol
  • Beta blocker drug

    J, Court DS (eds.). Medical Sciences. Elsevier Health Sciences. pp. 101–154 [150]. ISBN 978-0-7020-5249-1. Young R, Glennon RA (April 2009). "S(-)Propranolol

    Propranolol

    Propranolol

    Propranolol

  • Tetrodotoxin
  • Neurotoxin

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Tetrodotoxin

    Tetrodotoxin

    Tetrodotoxin

  • Amlodipine
  • Medication against high blood pressure

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Amlodipine

    Amlodipine

    Amlodipine

  • Meclizine
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Meclizine

    Meclizine

    Meclizine

  • Valproate
  • Medication used for epilepsy, bipolar disorder and migraine

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Valproate

    Valproate

    Valproate

  • Lamotrigine
  • Anticonvulsant medication

    review from South Asia". Indian Journal of Psychological Medicine. 37 (2): 154–158. doi:10.4103/0253-7176.155613. PMC 4418246. PMID 25969599. Wang S, Zheng

    Lamotrigine

    Lamotrigine

    Lamotrigine

  • Etripamil
  • Medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Etripamil

    Etripamil

  • Azetukalner
  • Experimental anticonvulsant

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Azetukalner

    Azetukalner

    Azetukalner

  • Crisugabalin
  • Drug for chronic pain

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Crisugabalin

    Crisugabalin

    Crisugabalin

  • Relutrigine
  • Pharmaceutical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Relutrigine

    Relutrigine

    Relutrigine

  • Minoxidil
  • Medication to treat high blood pressure and alopecia

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Minoxidil

    Minoxidil

    Minoxidil

  • Ranolazine
  • Drug used to treat angina

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Ranolazine

    Ranolazine

    Ranolazine

  • Phenytoin
  • Anti-seizure medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Phenytoin

    Phenytoin

    Phenytoin

  • Lidocaine
  • Local anesthetic

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Lidocaine

    Lidocaine

    Lidocaine

  • Sodium channel
  • Transmembrane protein allowing sodium ions in and out

    (2000). Principles of Neural Science (4th ed.). New York: McGraw-Hill. pp. 154–69. ISBN 978-0-8385-7701-1.{{cite book}}: CS1 maint: multiple names: authors

    Sodium channel

    Sodium channel

    Sodium_channel

  • Benzocaine
  • Local anaesthetic drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Benzocaine

    Benzocaine

    Benzocaine

  • Doxepin
  • Sedating antidepressant

    (3 and 6 mg) for the treatment of insomnia". Future Neurology. 6 (2): 143–154. doi:10.2217/fnl.10.83. ISSN 1479-6708. Dawkins K, Manji HK, Potter WZ (20

    Doxepin

    Doxepin

    Doxepin

  • Procaine
  • Local anesthetic drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Procaine

    Procaine

    Procaine

  • Oxcarbazepine
  • Anticonvulsant medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Oxcarbazepine

    Oxcarbazepine

    Oxcarbazepine

  • Baclofen
  • Muscle relaxant medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Baclofen

    Baclofen

    Baclofen

  • Lorazepam
  • Benzodiazepine medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Lorazepam

    Lorazepam

    Lorazepam

  • Flindokalner
  • Pharmaceutical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Flindokalner

    Flindokalner

    Flindokalner

  • Cholesterol
  • Sterol biosynthesized by all animal cells

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Cholesterol

    Cholesterol

    Cholesterol

  • Amiodarone
  • Antiarrhythmic medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Amiodarone

    Amiodarone

    Amiodarone

  • Dihydropyridine calcium channel blockers
  • Class of medication used to treat high blood pressure

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Dihydropyridine calcium channel blockers

    Dihydropyridine_calcium_channel_blockers

  • Buprenorphine
  • Opioid used to treat pain and opioid use disorder

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Buprenorphine

    Buprenorphine

    Buprenorphine

  • Voltage-gated sodium channel
  • Family of transport proteins

    extracellular immunoglobulin-like domain". The Journal of Cell Biology. 154 (2): 427–34. doi:10.1083/jcb.200102086. PMC 2150779. PMID 11470829. Antzelevitch

    Voltage-gated sodium channel

    Voltage-gated_sodium_channel

  • Diltiazem
  • Calcium channel blocker medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Diltiazem

    Diltiazem

    Diltiazem

  • Pregabalin
  • Anticonvulsant medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Pregabalin

    Pregabalin

    Pregabalin

  • Chlorzoxazone
  • Muscle relaxant

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Chlorzoxazone

    Chlorzoxazone

    Chlorzoxazone

  • Mirogabalin
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Mirogabalin

    Mirogabalin

    Mirogabalin

  • Topiramate
  • Medication used to treat epilepsy and migraine

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Topiramate

    Topiramate

    Topiramate

  • Sodium channel blocker
  • Several medications which disrupt the movement of Na+ ions

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Sodium channel blocker

    Sodium_channel_blocker

  • Erythromycin
  • Antibiotic medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Erythromycin

    Erythromycin

    Erythromycin

  • Calcium channel blocker
  • Drugs that disrupt movement of calcium across calcium channels

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Calcium channel blocker

    Calcium_channel_blocker

  • Atomoxetine
  • Medication used to treat ADHD

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Atomoxetine

    Atomoxetine

    Atomoxetine

  • Naminidil
  • Pharmaceutical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Naminidil

    Naminidil

    Naminidil

  • Gabapentin
  • Gamma-aminobutyric acid analog

    Cohort Study". Annals of Internal Medicine. 177 (Online ahead of print): 144–154. doi:10.7326/M23-0849. PMID 38224592. S2CID 266985259. Mersfelder TL, Nichols

    Gabapentin

    Gabapentin

    Gabapentin

  • Chlorphenamine
  • Antihistamine used to treat allergies

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Chlorphenamine

    Chlorphenamine

    Chlorphenamine

  • Nicardipine
  • Antihypertensive drug of the calcium channel blocker class

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Nicardipine

    Nicardipine

    Nicardipine

  • Flecainide
  • Antiarrhythmic medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Flecainide

    Flecainide

    Flecainide

  • Domperidone
  • Peripheral D2 receptor antagonist

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Domperidone

    Domperidone

    Domperidone

  • Diphenhydramine
  • Antihistamine medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Diphenhydramine

    Diphenhydramine

    Diphenhydramine

  • Solifenacin
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Solifenacin

    Solifenacin

    Solifenacin

  • Opakalim
  • Pharmaceutical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Opakalim

    Opakalim

    Opakalim

  • Licarbazepine
  • Active metabolite of oxcarbazepine

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Licarbazepine

    Licarbazepine

    Licarbazepine

  • Nifedipine
  • Calcium channel blocker medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Nifedipine

    Nifedipine

    Nifedipine

  • Glipizide
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Glipizide

    Glipizide

    Glipizide

  • Tamoxifen
  • Selective estrogen receptor modulator

    Estrogen/antiestrogen Action and Breast Cancer Therapy. Univ of Wisconsin Press. pp. 28, 154. ISBN 978-0-299-10480-1. Pratt WB (1994). The Anticancer Drugs. Oxford University

    Tamoxifen

    Tamoxifen

    Tamoxifen

  • Roxithromycin
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Roxithromycin

    Roxithromycin

    Roxithromycin

  • Barnidipine
  • Antihypertensive drug of the calcium channel blocker class

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Barnidipine

    Barnidipine

    Barnidipine

  • Bedaquiline
  • Medication used to treat tuberculosis

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Bedaquiline

    Bedaquiline

    Bedaquiline

  • Nortriptyline
  • Antidepressant medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Nortriptyline

    Nortriptyline

    Nortriptyline

  • Barbiturate
  • Class of depressant drugs derived from barbituric acid

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Barbiturate

    Barbiturate

    Barbiturate

  • Terfenadine
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Terfenadine

    Terfenadine

    Terfenadine

  • Lercanidipine
  • Antihypertensive drug of the calcium channel blocker class

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Lercanidipine

    Lercanidipine

    Lercanidipine

  • Cromakalim
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Cromakalim

    Cromakalim

    Cromakalim

  • Kava
  • Species of plant

    Revision) Variation—Australia New Zealand Food Standards Code – Amendment No. 154 - 2015-gs1906 - New Zealand Gazette". gazette.govt.nz. Archived from the

    Kava

    Kava

    Kava

  • Ion channel
  • Pore-forming membrane protein

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Ion channel

    Ion channel

    Ion_channel

  • Mexiletine
  • Pair of enantiomers

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Mexiletine

    Mexiletine

    Mexiletine

  • Fluoxakalner
  • Pharmaceutical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Fluoxakalner

    Fluoxakalner

    Fluoxakalner

  • PNU-282,987
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    PNU-282,987

    PNU-282,987

    PNU-282,987

  • Clarithromycin
  • Antibiotic medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Clarithromycin

    Clarithromycin

    Clarithromycin

  • Tolterodine
  • Benzhydryl compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Tolterodine

    Tolterodine

    Tolterodine

  • Safinamide
  • Reversible monoamine oxidase B inhibitor

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Safinamide

    Safinamide

    Safinamide

  • Piperocaine
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Piperocaine

    Piperocaine

    Piperocaine

  • Carbamazepine
  • Anticonvulsant medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Carbamazepine

    Carbamazepine

    Carbamazepine

  • Sotalol
  • Medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Sotalol

    Sotalol

    Sotalol

  • Pynegabine
  • Pharmaceutical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Pynegabine

    Pynegabine

    Pynegabine

  • Epithelial sodium channel blocker
  • (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Epithelial sodium channel blocker

    Epithelial sodium channel blocker

    Epithelial_sodium_channel_blocker

  • Channel opener
  • Index of articles associated with the same name

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Channel opener

    Channel_opener

  • Zonisamide
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Zonisamide

    Zonisamide

    Zonisamide

  • Tolperisone
  • Skeletal muscle relaxant drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Tolperisone

    Tolperisone

    Tolperisone

  • Isradipine
  • Antihypertensive drug of the calcium channel blocker class

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Isradipine

    Isradipine

    Isradipine

  • Amlodipine/celecoxib
  • Pain and blood pressure medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Amlodipine/celecoxib

    Amlodipine/celecoxib

  • Nicorandil
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Nicorandil

    Nicorandil

    Nicorandil

  • Mefenamic acid
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Mefenamic acid

    Mefenamic acid

    Mefenamic_acid

  • Bencyclane
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Bencyclane

    Bencyclane

    Bencyclane

  • Niguldipine
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Niguldipine

    Niguldipine

    Niguldipine

  • Nilvadipine
  • Antihypertensive drug of the calcium channel blocker class

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Nilvadipine

    Nilvadipine

    Nilvadipine

  • Saxitoxin
  • Paralytic shellfish toxin

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Saxitoxin

    Saxitoxin

    Saxitoxin

  • Cystic fibrosis transmembrane conductance regulator
  • Mammalian protein found in humans

    of the mammalian epididymis". Journal of Molecular Histology. 50 (2): 141–154. doi:10.1007/s10735-019-09813-3. PMID 30659401. S2CID 58026884. Sharma S

    Cystic fibrosis transmembrane conductance regulator

    Cystic fibrosis transmembrane conductance regulator

    Cystic_fibrosis_transmembrane_conductance_regulator

  • Arbaclofen placarbil
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Arbaclofen placarbil

    Arbaclofen placarbil

    Arbaclofen_placarbil

  • Encainide
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Encainide

    Encainide

    Encainide

  • Telmisartan/amlodipine/indapamide
  • Medication

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Telmisartan/amlodipine/indapamide

    Telmisartan/amlodipine/indapamide

  • Bay K8644
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Bay K8644

    Bay K8644

    Bay_K8644

  • 4-Methylpregabalin
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    4-Methylpregabalin

    4-Methylpregabalin

    4-Methylpregabalin

  • Pinacidil
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Pinacidil

    Pinacidil

    Pinacidil

  • Tetracaine
  • Local anaesthetic drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Tetracaine

    Tetracaine

    Tetracaine

  • Ziconotide
  • Drug for chronic pain

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Ziconotide

    Ziconotide

    Ziconotide

  • Pheneturide
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Pheneturide

    Pheneturide

    Pheneturide

  • Astemizole
  • Antihistamine drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Astemizole

    Astemizole

    Astemizole

  • Caroverine
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Caroverine

    Caroverine

    Caroverine

  • List of investigational antidepressants
  • List of pharmaceutical drugs under clinical development for treatment of depression

    TS-1211; TS-121) – vasopressin V1b receptor antagonist CB-03 (CB-04; CB-003; CB03-154) – KCNQ2 and KCNQ3 potassium channel stimulant Centanafadine (CTN; EB-1020)

    List of investigational antidepressants

    List_of_investigational_antidepressants

  • DSP-2230
  • Investigational analgesic drug

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    DSP-2230

    DSP-2230

    DSP-2230

  • Ketoconazole
  • Antifungal chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Ketoconazole

    Ketoconazole

    Ketoconazole

  • Gliclazide
  • Chemical compound

    (SsTx) XE-991 Activators KCNQ (Kv7)-specific: Azetukalner (encukalner) CB03-154 Fluoxakalner Flupirtine Opakalim Pynegabine Retigabine (ezogabine) IRKsTooltip

    Gliclazide

    Gliclazide

    Gliclazide

Searches for online references containing CB03 154

CB03 154

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CB03 154

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