Search references for RTIOX 276. Phrases containing RTIOX 276
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Orexin antagonist
RTIOX-276 is an orexin antagonist. RTIOX-276 binds selectively to the orexin 1 receptor (KE = 8.5nM) and lacks significant affinity for the orexin 2 receptor
RTIOX-276
Class of drugs
potential use in sleep disorders JNJ-10397049 – selective OX2 antagonist RTIOX-276 – selective OX1 antagonist SB-334867 – first non-peptide selective OX1
Orexin_antagonist
Pharmaceutical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Oveporexton
Medication used to treat insomnia
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Daridorexant
Neuropeptide that regulates arousal, wakefulness, and appetite
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Orexin
Pharmaceutical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Cleminorexton
Novel chemistry compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Alixorexton
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Lemborexant
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Firazorexton
Experimental anti-insomnia drug
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Seltorexant
G-protein-coupled receptor
Rocavorexant (C4X-3256; INDV-2000) – selective OX1 receptor antagonist RTIOX-276 – selective OX1 receptor antagonist SB-334867 – selective OX1 receptor
Orexin_receptor
Orexin receptor antagonist
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Fazamorexant
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Danavorexton
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Tebideutorexant
Medication used to treat insomnia
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Suvorexant
Protein-coding gene in the species Homo sapiens
Rocavorexant (C4X-3256; INDV-2000) - selective OX1 receptor antagonist RTIOX-276 - selective OX1 antagonist SB-334,867 - selective OX1 antagonist SB-408
Hypocretin (orexin) receptor 1
Hypocretin_(orexin)_receptor_1
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Vornorexant
Pharmaceutical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Ledasorexton
Stimulating neuropeptide
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Orexin-A
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
ACT-462206
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
ACT-335827
Pharmaceutical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Rocavorexant
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
JNJ-10397049
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
SB-334867
Orexin antagonist compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Almorexant
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
EMPA_(drug)
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
SB-649868
Protein-coding gene in the species Homo sapiens
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Hypocretin (orexin) receptor 2
Hypocretin_(orexin)_receptor_2
Antagonists: ACT-335827 ACT-462206 Almorexant Filorexant Lemborexant Nemorexant RTIOX-276 SB-334867 SB-408124 SB-649868 Suvorexant TCS-1102 Agonists: Orexin (A
List of signaling peptide/protein receptor modulators
List_of_signaling_peptide/protein_receptor_modulators
Pharmaceutical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Balumorexton
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Suntinorexton
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Filorexant
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
Nivasorexant
Chemical compound
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
SB-408124
Orexin antagonist
Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)
TCS-OX2-29
RTIOX 276
RTIOX 276
RTIOX 276
RTIOX 276
Boy/Male
Muslim/Islamic
Belief
Boy/Male
Hindu
Resembling a God, Poet
Girl/Female
Australian, Greek, Irish
Prophetess
Male
Iranian/Persian
Contracted form of Persian Dârayavahush, DARAWESH means "possesses a lot; wealthy."
Boy/Male
Sikh
Bravely upholding the truth, Achiever
Boy/Male
Irish
Peace from God.
Girl/Female
Indian
Star, Beautiful
Female
Hebrew
 Variant spelling of Hebrew unisex Rinnah, RINA means "shouting for joy." Compare with other forms of Rina.
Girl/Female
Indian
Rain, Constant flow
Boy/Male
Hindu, Indian, Traditional
Lord of Empire
RTIOX 276
RTIOX 276
RTIOX 276
RTIOX 276
RTIOX 276