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RTIOX 276

  • RTIOX-276
  • Orexin antagonist

    RTIOX-276 is an orexin antagonist. RTIOX-276 binds selectively to the orexin 1 receptor (KE = 8.5nM) and lacks significant affinity for the orexin 2 receptor

    RTIOX-276

    RTIOX-276

    RTIOX-276

  • Orexin antagonist
  • Class of drugs

    potential use in sleep disorders JNJ-10397049 – selective OX2 antagonist RTIOX-276 – selective OX1 antagonist SB-334867 – first non-peptide selective OX1

    Orexin antagonist

    Orexin_antagonist

  • Oveporexton
  • Pharmaceutical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Oveporexton

    Oveporexton

    Oveporexton

  • Daridorexant
  • Medication used to treat insomnia

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Daridorexant

    Daridorexant

    Daridorexant

  • Orexin
  • Neuropeptide that regulates arousal, wakefulness, and appetite

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Orexin

    Orexin

    Orexin

  • Cleminorexton
  • Pharmaceutical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Cleminorexton

    Cleminorexton

    Cleminorexton

  • Alixorexton
  • Novel chemistry compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Alixorexton

    Alixorexton

    Alixorexton

  • Lemborexant
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Lemborexant

    Lemborexant

    Lemborexant

  • Firazorexton
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Firazorexton

    Firazorexton

    Firazorexton

  • Seltorexant
  • Experimental anti-insomnia drug

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Seltorexant

    Seltorexant

    Seltorexant

  • Orexin receptor
  • G-protein-coupled receptor

    Rocavorexant (C4X-3256; INDV-2000) – selective OX1 receptor antagonist RTIOX-276 – selective OX1 receptor antagonist SB-334867 – selective OX1 receptor

    Orexin receptor

    Orexin_receptor

  • Fazamorexant
  • Orexin receptor antagonist

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Fazamorexant

    Fazamorexant

    Fazamorexant

  • Danavorexton
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Danavorexton

    Danavorexton

    Danavorexton

  • Tebideutorexant
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Tebideutorexant

    Tebideutorexant

    Tebideutorexant

  • Suvorexant
  • Medication used to treat insomnia

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Suvorexant

    Suvorexant

    Suvorexant

  • Hypocretin (orexin) receptor 1
  • Protein-coding gene in the species Homo sapiens

    Rocavorexant (C4X-3256; INDV-2000) - selective OX1 receptor antagonist RTIOX-276 - selective OX1 antagonist SB-334,867 - selective OX1 antagonist SB-408

    Hypocretin (orexin) receptor 1

    Hypocretin (orexin) receptor 1

    Hypocretin_(orexin)_receptor_1

  • Vornorexant
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Vornorexant

    Vornorexant

    Vornorexant

  • Ledasorexton
  • Pharmaceutical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Ledasorexton

    Ledasorexton

    Ledasorexton

  • Orexin-A
  • Stimulating neuropeptide

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Orexin-A

    Orexin-A

  • ACT-462206
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    ACT-462206

    ACT-462206

    ACT-462206

  • ACT-335827
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    ACT-335827

    ACT-335827

    ACT-335827

  • Rocavorexant
  • Pharmaceutical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Rocavorexant

    Rocavorexant

    Rocavorexant

  • JNJ-10397049
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    JNJ-10397049

    JNJ-10397049

    JNJ-10397049

  • SB-334867
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    SB-334867

    SB-334867

    SB-334867

  • Almorexant
  • Orexin antagonist compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Almorexant

    Almorexant

    Almorexant

  • EMPA (drug)
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    EMPA (drug)

    EMPA (drug)

    EMPA_(drug)

  • SB-649868
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    SB-649868

    SB-649868

    SB-649868

  • Hypocretin (orexin) receptor 2
  • Protein-coding gene in the species Homo sapiens

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Hypocretin (orexin) receptor 2

    Hypocretin (orexin) receptor 2

    Hypocretin_(orexin)_receptor_2

  • List of signaling peptide/protein receptor modulators
  • Antagonists: ACT-335827 ACT-462206 Almorexant Filorexant Lemborexant Nemorexant RTIOX-276 SB-334867 SB-408124 SB-649868 Suvorexant TCS-1102 Agonists: Orexin (A

    List of signaling peptide/protein receptor modulators

    List_of_signaling_peptide/protein_receptor_modulators

  • Balumorexton
  • Pharmaceutical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Balumorexton

    Balumorexton

    Balumorexton

  • Suntinorexton
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Suntinorexton

    Suntinorexton

    Suntinorexton

  • Filorexant
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Filorexant

    Filorexant

    Filorexant

  • Nivasorexant
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    Nivasorexant

    Nivasorexant

    Nivasorexant

  • SB-408124
  • Chemical compound

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    SB-408124

    SB-408124

    SB-408124

  • TCS-OX2-29
  • Orexin antagonist

    Lemborexant Nivasorexant (ACT-539313) Rocavorexant (C4X-3256; INDV-2000 RTIOX-276 SB-334867 SB-408124 Suvorexant TCS-1102 Tebideutorexant (JNJ-61393215)

    TCS-OX2-29

    TCS-OX2-29

    TCS-OX2-29

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RTIOX 276

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RTIOX 276

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RTIOX 276

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RTIOX 276

Online names & meanings

  • Yaqeen
  • Boy/Male

    Muslim/Islamic

    Yaqeen

    Belief

  • Devin
  • Boy/Male

    Hindu

    Devin

    Resembling a God, Poet

  • Sibeal
  • Girl/Female

    Australian, Greek, Irish

    Sibeal

    Prophetess

  • DARAWESH
  • Male

    Iranian/Persian

    DARAWESH

    Contracted form of Persian Dârayavahush, DARAWESH means "possesses a lot; wealthy."

  • Sadipak
  • Boy/Male

    Sikh

    Sadipak

    Bravely upholding the truth, Achiever

  • Gorry
  • Boy/Male

    Irish

    Gorry

    Peace from God.

  • Najmah
  • Girl/Female

    Indian

    Najmah

    Star, Beautiful

  • RINA
  • Female

    Hebrew

    RINA

     Variant spelling of Hebrew unisex Rinnah, RINA means "shouting for joy." Compare with other forms of Rina.

  • Dhara
  • Girl/Female

    Indian

    Dhara

    Rain, Constant flow

  • Takhvinder
  • Boy/Male

    Hindu, Indian, Traditional

    Takhvinder

    Lord of Empire

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RTIOX 276

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RTIOX 276

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RTIOX 276

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RTIOX 276