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PPAR AGONIST

  • PPAR agonist
  • Drug used for the treatment of symptoms of metabolic syndrome

    PPAR agonists are drugs which act upon the peroxisome proliferator-activated receptor. They are used for the treatment of symptoms of the metabolic syndrome

    PPAR agonist

    PPAR agonist

    PPAR_agonist

  • Lanifibranor
  • Chemical compound

    proliferator-activated receptor (PPAR) agonist and is the first medication that targets PPAR-alpha, PPAR-beta, and PPAR-gamma simultaneously. As of 2023

    Lanifibranor

    Lanifibranor

    Lanifibranor

  • Peroxisome proliferator-activated receptor
  • Group of nuclear receptor proteins

    Malaguarnera R (2009). "PPAR-gamma Agonists and Their Effects on IGF-I Receptor Signaling: Implications for Cancer". PPAR Res. 2009 830501. doi:10.1155/2009/830501

    Peroxisome proliferator-activated receptor

    Peroxisome proliferator-activated receptor

    Peroxisome_proliferator-activated_receptor

  • Retatrutide
  • Chemical compound

    pharmaceutical company Eli Lilly and Company. It is a triple hormone receptor agonist on the GLP-1, GIP, and glucagon receptors. The safety profile of retatrutide

    Retatrutide

    Retatrutide

    Retatrutide

  • Drug class
  • Group of similar medications

    (atherosclerosis). However, not all PPAR agonists are fibrates, not all triglyceride-lowering agents are PPAR agonists, and not all drugs used to treat atherosclerosis

    Drug class

    Drug_class

  • Tianeptine
  • Atypical antidepressant

    (R)-Tianeptine is a weak μ-opioid receptor agonist, while estianeptine is a peroxisome proliferator-activated receptor (PPAR) agonist. Although several related compounds

    Tianeptine

    Tianeptine

    Tianeptine

  • Saroglitazar
  • Chemical compound

    acts as a dual PPAR agonist at the subtypes α (alpha) and γ (gamma) of the peroxisome proliferator-activated receptor (PPAR). Agonist action on PPARα

    Saroglitazar

    Saroglitazar

    Saroglitazar

  • Orforglipron
  • Anti-obesity medication

    name Foundayo, is an oral, non-peptide, small-molecule GLP-1 receptor agonist developed as a weight loss drug by Eli Lilly and Company. It was discovered

    Orforglipron

    Orforglipron

    Orforglipron

  • Empagliflozin
  • Diabetes medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Empagliflozin

    Empagliflozin

  • Tirzepatide
  • Anti-diabetic and anti-obesity medication

    is a gastric inhibitory polypeptide (GIP) analog and a GLP-1 receptor agonist. It is used as an antidiabetic medication to treat type 2 diabetes (T2D)

    Tirzepatide

    Tirzepatide

    Tirzepatide

  • Elafibranor
  • Chemical compound

    dual PPARα/δ agonist. Elafibranor and its main active metabolite GFT1007 are peroxisome proliferator-activated receptor (PPAR) agonists, both of which

    Elafibranor

    Elafibranor

    Elafibranor

  • Semaglutide
  • Anti-diabetic and anti-obesity medication

    peptide-1 (GLP-1), modified with a side chain, and acts as a GLP-1 receptor agonist. The most common side effects include nausea, vomiting, diarrhea, abdominal

    Semaglutide

    Semaglutide

    Semaglutide

  • GLP1 poly-agonist peptides
  • Class of drugs used to treat diabetes

    GLP1 poly-agonist peptides are a class of drugs that activate multiple peptide hormone receptors including the glucagon-like peptide-1 (GLP-1) receptor

    GLP1 poly-agonist peptides

    GLP1_poly-agonist_peptides

  • Survodutide
  • Peptide drug

    peptide that works as a dual glucagon/GLP-1 receptor agonist. Unlike other dual GLP-1/glucagon dual agonists, it is a glucagon analog rather than an analog

    Survodutide

    Survodutide

    Survodutide

  • Liraglutide
  • Anti-diabetic medication

    the skin. Liraglutide is a glucagon-like peptide-1 receptor agonist (GLP-1 receptor agonist) also known as incretin mimetics. It works by increasing insulin

    Liraglutide

    Liraglutide

    Liraglutide

  • Estianeptine
  • Pharmaceutical compound

    code name TNX-4300, is a peroxisome proliferator-activated receptor (PPAR) agonist and atypical tricyclic antidepressant (TCA) which is under development

    Estianeptine

    Estianeptine

    Estianeptine

  • Glucagon-like peptide-1
  • Gastrointestinal peptide hormone involved in glucose homeostasis

    preserved in patients with type 2 diabetes. Glucagon-like peptide-1 receptor agonists gained approval as drugs to treat diabetes and obesity starting in the

    Glucagon-like peptide-1

    Glucagon-like peptide-1

    Glucagon-like_peptide-1

  • Biguanide
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Biguanide

    Biguanide

    Biguanide

  • Telmisartan
  • Blood pressure medication

    renin–angiotensin system, telmisartan acts as a partial agonist of peroxisome proliferator-activated receptor gamma (PPAR-γ), a central regulator of insulin and glucose

    Telmisartan

    Telmisartan

    Telmisartan

  • Danuglipron
  • Chemical compound

    Danuglipron is a small-molecule GLP-1 receptor agonist, formerly under development by Pfizer that, in an oral formulation, was under investigation as

    Danuglipron

    Danuglipron

    Danuglipron

  • Dulaglutide
  • Diabetes medication

    incretin mimetics, as it is a glucagon-like peptide-1 receptor agonist (GLP-1 agonist) consisting of GLP-1(7-37) covalently linked to an Fc fragment of

    Dulaglutide

    Dulaglutide

    Dulaglutide

  • GW501516
  • Abandoned metabolic and cardiovascular drug

    Newsholme SJ (2009). PS 895 - Rat carcinogenicity study with GW501516, a PPAR delta agonist (PDF). 48th Annual Meeting of the Society of Toxicology. Baltimore:

    GW501516

    GW501516

    GW501516

  • Insulin glargine
  • Long-acting insulin

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin glargine

    Insulin glargine

    Insulin_glargine

  • Dapagliflozin
  • Diabetes medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Dapagliflozin

    Dapagliflozin

    Dapagliflozin

  • Sitagliptin
  • Diabetes medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Sitagliptin

    Sitagliptin

    Sitagliptin

  • Sitagliptin/metformin
  • Pharmaceutical drug

    combination therapy with a peroxisome proliferator-activated receptor (PPAR) agonist (i.e., a thiazolidinedione) as an adjunct to diet and exercise in people

    Sitagliptin/metformin

    Sitagliptin/metformin

  • Brenipatide
  • Pharmaceutical compound

    United States Adopted Name; developmental code name LY-3537031) is a dual agonist of glucagon-like peptide-1 (GLP-1) receptors and gastric inhibitory polypeptide

    Brenipatide

    Brenipatide

  • Alpha agonist
  • Topics referred to by the same term

    Alpha agonist may refer to: Alpha-adrenergic agonist, drugs that selectively stimulate alpha adrenergic receptors PPAR-alpha agonist, drugs which act upon

    Alpha agonist

    Alpha_agonist

  • Insulin efsitora alfa
  • Medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin efsitora alfa

    Insulin_efsitora_alfa

  • Peroxisome proliferator-activated receptor delta
  • Nuclear receptor protein found in humans

    increase in type I fibers. Both PPAR-delta and AMPK agonists are regarded as exercise mimetics. In adipose tissue PPAR-β/δ increases both oxidation as

    Peroxisome proliferator-activated receptor delta

    Peroxisome proliferator-activated receptor delta

    Peroxisome_proliferator-activated_receptor_delta

  • SGLT2 inhibitor
  • Class of medication

    systematic review and network meta-analysis comparing SGLT-2 inhibitors, GLP-1 agonists, and DPP-4 inhibitors demonstrated that use of SGLT2 inhibitors was associated

    SGLT2 inhibitor

    SGLT2_inhibitor

  • Canagliflozin
  • Chemical compound

    Study of Diabetes consider either a SGLT2 inhibitor or GLP-1 receptor agonist a reasonable second line medication in those with heart disease. Canagliflozin

    Canagliflozin

    Canagliflozin

    Canagliflozin

  • Sulfonylurea
  • Class of organic compounds used in medicine and agriculture

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Sulfonylurea

    Sulfonylurea

    Sulfonylurea

  • Chiglitazar
  • Chemical compound

    type 2 diabetes. It is a peroxisome proliferator-activated receptor (PPAR) agonist. In China, chiglitazar is approved for glycemic control in adult patients

    Chiglitazar

    Chiglitazar

    Chiglitazar

  • Metformin
  • Medication used to treat diabetes

    conclusive evidence of improved live birth rates was found. In long GnRH-agonist protocols there was uncertainty in the evidence of improved live birth

    Metformin

    Metformin

    Metformin

  • Diabetes medication
  • Drugs that lower blood glucose levels to treat diabetes

    mellitus by decreasing glucose levels in the blood. Most GLP-1 receptor agonists (liraglutide, exenatide, tirzepatide, pramlintide and others) are administered

    Diabetes medication

    Diabetes_medication

  • Insulin analogue
  • Modified forms of synthetic insulin

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin analogue

    Insulin analogue

    Insulin_analogue

  • Dipeptidyl peptidase-4 inhibitor
  • Enzyme blocker and diabetes treatment drug

    of Sodium-Glucose Cotransporter 2 Inhibitors, Glucagon-like Peptide 1 Agonists, and Dipeptidyl Peptidase 4 Inhibitors With All-Cause Mortality in Patients

    Dipeptidyl peptidase-4 inhibitor

    Dipeptidyl peptidase-4 inhibitor

    Dipeptidyl_peptidase-4_inhibitor

  • List of commercially available insulins
  • consistently, allowing for prolonged action. Liraglutide, a GLP-1 receptor agonist, mimics the effects of incretin hormones by enhancing insulin secretion

    List of commercially available insulins

    List of commercially available insulins

    List_of_commercially_available_insulins

  • Mazdutide
  • GLP1 poly-agonist drug

    Mazdutide (also known as IBI362 or LY3305677) is a dual agonist of the GLP-1 receptor and glucagon receptor. It is an analog of oxyntomodulin (OXM). The

    Mazdutide

    Mazdutide

  • GW0742
  • PPAR β/δ receptor Agonist compound

    and fitorine) is a PPARδ/β agonist that has been investigated for drug use by GlaxoSmithKline. It is mixed PPAR-B agonist antagonist depending on its

    GW0742

    GW0742

    GW0742

  • Vildagliptin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Vildagliptin

    Vildagliptin

    Vildagliptin

  • Pioglitazone
  • Chemical compound

    receptor peroxisome proliferator-activated receptor gamma (PPAR-γ) and to a lesser extent PPAR-α. It modulates the transcription of the genes involved in

    Pioglitazone

    Pioglitazone

    Pioglitazone

  • Seladelpar
  • Chemical compound

    February 2025. Retrieved 27 February 2025. Billin AN (October 2008). "PPAR-beta/delta agonists for Type 2 diabetes and dyslipidemia: an adopted orphan still looking

    Seladelpar

    Seladelpar

    Seladelpar

  • Thiazolidinedione
  • Class of chemical compounds

    specific for PPARγ (PPAR-gamma, PPARG). They are thus the PPARG agonists subset of PPAR agonists. The endogenous ligands for these receptors are free fatty

    Thiazolidinedione

    Thiazolidinedione

    Thiazolidinedione

  • Acarbose
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Acarbose

    Acarbose

    Acarbose

  • Abrine
  • Chemical compound

    Chen, Calvin Yu-Chian (2014). "In Silico Identification of Potent PPAR-γ Agonists from Traditional Chinese Medicine: A Bioactivity Prediction, Virtual

    Abrine

    Abrine

    Abrine

  • Aleglitazar
  • Chemical compound

    Aleglitazar is a peroxisome proliferator-activated receptor agonist (hence a PPAR modulator) with affinity to PPARα and PPARγ, which was under development

    Aleglitazar

    Aleglitazar

    Aleglitazar

  • Insulin aspart
  • Rapid-acting man-made insulin

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin aspart

    Insulin aspart

    Insulin_aspart

  • NPH insulin
  • Intermediate acting insulin formulation

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    NPH insulin

    NPH insulin

    NPH_insulin

  • Peroxisome proliferator-activated receptor alpha
  • Nuclear receptor protein found in humans

    contrast to statins. PPAR-α, agonists may carry therapeutic value for the treatment of non-alcoholic fatty liver disease. PPAR-alpha may also be a site

    Peroxisome proliferator-activated receptor alpha

    Peroxisome proliferator-activated receptor alpha

    Peroxisome_proliferator-activated_receptor_alpha

  • Peroxisome proliferator-activated receptor gamma
  • Nuclear receptor protein found in humans

    genes. Three subtypes of PPARs are known: PPAR-alpha, PPAR-delta, and PPAR-gamma. The protein encoded by this gene is PPAR-gamma and is a regulator of

    Peroxisome proliferator-activated receptor gamma

    Peroxisome proliferator-activated receptor gamma

    Peroxisome_proliferator-activated_receptor_gamma

  • Insulin lispro
  • Rapid-acting insuline analog

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin lispro

    Insulin lispro

    Insulin_lispro

  • Insulin icodec
  • Ultralong-acting basal insulin analogue

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin icodec

    Insulin_icodec

  • Bisphenol A diglycidyl ether
  • Chemical compound

    v t e Androgen receptor modulators ARTooltip Androgen receptor Agonists Testosterone derivatives: 4-Androstenediol 4-Dehydroepiandrosterone (4-DHEA)

    Bisphenol A diglycidyl ether

    Bisphenol A diglycidyl ether

    Bisphenol_A_diglycidyl_ether

  • Rosiglitazone
  • Chemical compound

    thiazolidinedione class. It works as an insulin sensitizer, by binding to the PPAR in fat cells and making the cells more responsive to insulin. It is marketed

    Rosiglitazone

    Rosiglitazone

    Rosiglitazone

  • Insulin degludec
  • Ultralong-acting basal insulin analogue

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin degludec

    Insulin degludec

    Insulin_degludec

  • Selective PPAR modulator
  • SPPARMs of the PPARγ, BADGE, EPI-001, INT-131, MK-0533, and S26948. PPAR agonist Fruchart, Jean-Charles; Santos, Raul D.; Aguilar-Salinas, Carlos; Aikawa

    Selective PPAR modulator

    Selective_PPAR_modulator

  • Linagliptin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Linagliptin

    Linagliptin

    Linagliptin

  • EPI-001
  • Chemical compound

    (incl. AASTooltip anabolic–androgenic steroid) ARTooltip Androgen receptor agonists Testosterone derivatives: Androstenediol dipropionate Boldenone undecylenate

    EPI-001

    EPI-001

  • Exenatide
  • Medication

    unclear safety. Exenatide is a glucagon-like peptide-1 receptor agonist (GLP-1 receptor agonist) also known as incretin mimetics. It works by increasing insulin

    Exenatide

    Exenatide

    Exenatide

  • Gliclazide
  • Chemical compound

    caused by danazol, chlorpromazine, glucocorticoids, progestogens, or β-2 agonists. Its hypoglycemic action may be potentiated by phenylbutazone, alcohol

    Gliclazide

    Gliclazide

    Gliclazide

  • Glipizide
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Glipizide

    Glipizide

    Glipizide

  • Glibenclamide
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Glibenclamide

    Glibenclamide

    Glibenclamide

  • Troglitazone
  • Chemical compound

    moiety, potentially giving it vitamin E-like activity in addition to its PPAR activation. It has been shown to reduce inflammation. Troglitazone use was

    Troglitazone

    Troglitazone

    Troglitazone

  • Dasiglucagon
  • Medication

    operates through the same mechanism as endogenous glucagon, acting as an agonist at glucagon receptors expressed throughout the body, which are G-coupled

    Dasiglucagon

    Dasiglucagon

  • Tesaglitazar
  • Chemical compound

    known as AZ 242) is a dual peroxisome proliferator-activated receptor agonist with affinity to PPARα and PPARγ, proposed for the management of type 2

    Tesaglitazar

    Tesaglitazar

    Tesaglitazar

  • Alogliptin
  • Anti-diabetic drug

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Alogliptin

    Alogliptin

    Alogliptin

  • Fenofibrate/pravastatin
  • Combination medication

    enzymes. Fenofibrate is a peroxisome proliferator-activated receptor (PPAR) agonist. It activates a type of receptor called the peroxisome proliferator-activated

    Fenofibrate/pravastatin

    Fenofibrate/pravastatin

  • Primary biliary cholangitis
  • Autoimmune disease of the liver

    2024. Elafibranor is a peroxisome proliferator-activated receptor (PPAR) agonist, and while the mechanism of action is not fully understood, it is thought

    Primary biliary cholangitis

    Primary biliary cholangitis

    Primary_biliary_cholangitis

  • Ertugliflozin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Ertugliflozin

    Ertugliflozin

    Ertugliflozin

  • Bexagliflozin
  • Antidiabetic medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Bexagliflozin

    Bexagliflozin

  • Dapagliflozin/sitagliptin
  • Medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Dapagliflozin/sitagliptin

    Dapagliflozin/sitagliptin

  • Lotiglipron
  • Chemical compound

    Lotiglipron is a non-peptide GLP-1 receptor agonist which was under development by Pfizer as a weight loss drug. However, it was withdrawn from development

    Lotiglipron

    Lotiglipron

    Lotiglipron

  • Empagliflozin/linagliptin/metformin
  • Combination drug

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Empagliflozin/linagliptin/metformin

    Empagliflozin/linagliptin/metformin

  • Glimepiride
  • Medication

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Glimepiride

    Glimepiride

    Glimepiride

  • Sodelglitazar
  • Chemical compound

    PPARδ receptor agonist developed by GlaxoSmithKline. While it is primarily active at the PPARδ receptor, it is considered a pan agonist with activity at

    Sodelglitazar

    Sodelglitazar

    Sodelglitazar

  • Conveglipron
  • Pharmaceutical compound

    developmental code name HDM1002) is a glucagon-like peptide-1 (GLP-1) receptor agonist which is under development for the treatment of type 2 diabetes, obesity

    Conveglipron

    Conveglipron

    Conveglipron

  • Gemigliptin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Gemigliptin

    Gemigliptin

    Gemigliptin

  • Glibenclamide/metformin
  • Combination drug

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Glibenclamide/metformin

    Glibenclamide/metformin

  • Lixisenatide
  • Diabetes drug

    and manufactured by Sanofi) is a once-daily injectable GLP-1 receptor agonist for the treatment of type 2 diabetes. Lixisenatide is used as adjunct to

    Lixisenatide

    Lixisenatide

    Lixisenatide

  • Lobeglitazone
  • Chemical compound

    thiazolidinedione class of drugs. As an agonist for both PPARα and PPARγ, it works as an insulin sensitizer by binding to the PPAR receptors in fat cells and making

    Lobeglitazone

    Lobeglitazone

  • Insulin (medication)
  • Use of insulin protein and analogs as medical treatment

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin (medication)

    Insulin (medication)

    Insulin_(medication)

  • Sotagliflozin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Sotagliflozin

    Sotagliflozin

  • Vildagliptin/metformin
  • Pharmaceutical drug

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Vildagliptin/metformin

    Vildagliptin/metformin

  • Insulin glargine/lixisenatide
  • Combination drug

    American Diabetes Association, combination treatment of a GLP-1 receptor agonist with basal insulin should occur after HbA1C levels remain above target

    Insulin glargine/lixisenatide

    Insulin_glargine/lixisenatide

  • Regular insulin
  • Short-acting insulin formulation

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Regular insulin

    Regular insulin

    Regular_insulin

  • Voglibose
  • Alpha-glucosidase inhibitor

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Voglibose

    Voglibose

    Voglibose

  • Tofogliflozin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Tofogliflozin

    Tofogliflozin

    Tofogliflozin

  • Insulin detemir
  • Long-acting man-made insulin

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Insulin detemir

    Insulin_detemir

  • Dapagliflozin/metformin
  • Two drugs combined to treat diabetes

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Dapagliflozin/metformin

    Dapagliflozin/metformin

  • Repaglinide
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Repaglinide

    Repaglinide

    Repaglinide

  • Alpha-glucosidase inhibitor
  • Oral anti-diabetic drugs

    Therapy: Metformin, Alpha-Glucosidase Inhibitors, Pioglitazone, GLP-1 Agonists, DPP-IV Inhibitors, and SGLT-2 Inhibitors. Michelle DeGeeter, PharmD, CDE

    Alpha-glucosidase inhibitor

    Alpha-glucosidase_inhibitor

  • Tetradecylthioacetic acid
  • Chemical compound

    dyslipidaemia in male patients with type 2 diabetes mellitus, possibly by dual PPAR-alpha/delta activation and increased mitochondrial fatty acid oxidation"

    Tetradecylthioacetic acid

    Tetradecylthioacetic_acid

  • Imeglimin
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Imeglimin

    Imeglimin

    Imeglimin

  • Meglitinide
  • Chemical substance

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Meglitinide

    Meglitinide

    Meglitinide

  • Glisoxepide
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Glisoxepide

    Glisoxepide

    Glisoxepide

  • Remogliflozin etabonate
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Remogliflozin etabonate

    Remogliflozin etabonate

    Remogliflozin_etabonate

  • Empagliflozin/metformin
  • Pharmaceutical drug

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Empagliflozin/metformin

    Empagliflozin/metformin

  • Miglitol
  • Chemical compound

    PPAR agonists Ciglitazone§ Darglitazone§ Englitazone§ Lobeglitazone Netoglitazone§ Pioglitazone Rivoglitazone† Rosiglitazone Troglitazone‡ Dual PPAR agonists

    Miglitol

    Miglitol

    Miglitol

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  • Premveer
  • Boy/Male

    Sikh

    Premveer

    Pyar ko pasand karne wala

    Premveer

  • Perye
  • Boy/Male

    American, British, English

    Perye

    From the Pear Tree

    Perye

  • DurEShahwar
  • Girl/Female

    Arabic, Muslim

    DurEShahwar

    Kings Worthy Pear

    DurEShahwar

  • Aadamya
  • Boy/Male

    Indian

    Aadamya

    Apne Dam par

    Aadamya

  • Hrusosky
  • Boy/Male

    Czechoslovakian

    Hrusosky

    Dwells near the pear tree.

    Hrusosky

  • Peri
  • Girl/Female

    Australian, British, English, German, Greek, Hebrew

    Peri

    Female Version of Perry; Pear Tree

    Peri

  • Pear
  • Surname or Lastname

    English

    Pear

    English : from Middle English pe(e)re ‘pear’ (Old English pere, peru, from Latin pirum), a metonymic occupational name for a grower or seller of pears, or a topographic name for someone who lived by a pear tree or pear orchard.English : nickname from Middle English pere ‘peer’, ‘companion’ (Old French pe(e)r, from Latin par ‘equal’).Jewish : Americanization of some like-sounding Ashkenazic surname; e.g. possibly a shortened form of a surname such as Pearl, Pearlman, or Pearlstein.

    Pear

  • BELIT
  • Female

    Babylonian

    BELIT

    , ("the lady"), par excellence.

    BELIT

  • Apar
  • Boy/Male

    Hindu

    Apar

    Limitless

    Apar

  • Aadamya | ஆதம்ய
  • Boy/Male

    Tamil

    Aadamya | ஆதம்ய

    Apne Dam par

    Aadamya | ஆதம்ய

  • Perri
  • Boy/Male

    Australian, British, English, French

    Perri

    Wanderer; Pear Tree

    Perri

  • Perry
  • Boy/Male

    Christian & English(British/American/Australian)

    Perry

    Pear Tree

    Perry

  • Pyar
  • Girl/Female

    Indian, Punjabi, Sikh

    Pyar

    Love

    Pyar

  • Apar
  • Boy/Male

    Hindu, Indian, Punjabi

    Apar

    Infinite; Great; Best; Endless

    Apar

  • BELTIS
  • Female

    Babylonian

    BELTIS

    , ("the lady"), par excellence.

    BELTIS

  • Perrie
  • Girl/Female

    Australian, French

    Perrie

    Pear Tree

    Perrie

  • Perrie
  • Boy/Male

    British, English

    Perrie

    From the Pear Tree

    Perrie

  • Peare
  • Surname or Lastname

    English

    Peare

    English : variant spelling of Pear.

    Peare

  • Perry
  • Girl/Female

    Australian, British, English, French, German

    Perry

    Pear Tree

    Perry

  • Piar
  • Boy/Male

    Indian, Punjabi, Sikh

    Piar

    Love; Affection

    Piar

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PPAR AGONIST

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PPAR AGONIST

  • Pear-shaped
  • a.

    Of the form of a pear.

  • Pear
  • n.

    The fleshy pome, or fruit, of a rosaceous tree (Pyrus communis), cultivated in many varieties in temperate climates; also, the tree which bears this fruit. See Pear family, below.

  • Pyriform
  • a.

    Having the form of a pear; pear-shaped.

  • Spathiform
  • a.

    Resembling spar in form.

  • Bergamot
  • n.

    A variety of pear.

  • Shiver-spar
  • n.

    A variety of calcite, so called from its slaty structure; -- called also slate spar.

  • Sparring
  • p. pr. & vb. n.

    of Spar

  • Pery
  • n.

    A pear tree. See Pirie.

  • Spar-hung
  • a.

    Hung with spar, as a cave.

  • Pirie
  • n.

    A pear tree.

  • Sparry
  • a.

    Resembling spar, or consisting of spar; abounding with spar; having a confused crystalline structure; spathose.

  • Sparred
  • imp. & p. p.

    of Spar

  • Perjenet
  • n.

    A kind of pear.

  • Cand
  • n.

    Fluor spar. See Kand.

  • Tolypeutine
  • n.

    The apar.

  • Spar
  • n.

    An old name for a nonmetallic mineral, usually cleavable and somewhat lustrous; as, calc spar, or calcite, fluor spar, etc. It was especially used in the case of the gangue minerals of a metalliferous vein.

  • Muscadine
  • n.

    A fragrant and delicious pear.

  • Par
  • prep.

    By; with; -- used frequently in Early English in phrases taken from the French, being sometimes written as a part of the word which it governs; as, par amour, or paramour; par cas, or parcase; par fay, or parfay.