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Chemical compound
Nepadutant (INN; development code MEN-11420) is a glycosylated bicyclic cyclohexapeptide drug which acts as a highly selective NK2 receptor antagonist
Nepadutant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Elinzanetant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Fezolinetant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Tradipitant
Veterinary medication
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Maropitant
Chemical compound (polypeptide neurotransmitter)
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Substance_P
Protein-coding gene in the species Homo sapiens
Phase 3 trial results in 2009, and abandoned by Sanofi-Aventis GR-159897 Nepadutant MEN-10376 - potent and selective antagonist, 7-amino acid polypeptide
Tachykinin_receptor_2
Protein family
tachykinin antagonists include: Aprepitant Casopitant Fosaprepitant Maropitant Nepadutant Osanetant Saredutant Talnetant Tachykinin InterPro: IPR008215 Grace RC
Tachykinin_peptides
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Aprepitant
Chemical compound class
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
NK1_receptor_antagonist
Pharmaceutical drug
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Netupitant/palonosetron
Pharmaceutical drug
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Rolapitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Netupitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Fosaprepitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Pavinetant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Osanetant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Ezlopitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Vestipitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Neurokinin_B
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Neurokinin_A
Protein-coding gene in the species Homo sapiens
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Tachykinin_receptor_1
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Casopitant
Chemical compound
for the treatment of major depressive disorder. GR-159,897 Ibodutant Nepadutant Hopkins CR (October 2010). "ACS chemical neuroscience molecule spotlight
Saredutant
Protein-coding gene in the species Homo sapiens
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Tachykinin_receptor_3
Neosar Neoscan Neosporin neostigmine bromide (INN) Neothylline Neotrizine nepadutant (INN) nepafenac (INN) nepaprazole (INN) Nephramine 5.4% Nephroflow nepicastat
List_of_drugs:_Nb–Nh
Chemical compound
because of low response and negative results of study NAK-06. GR-159,897 Nepadutant Saredutant "Clinical Trials Database". Menarini Group. Retrieved 11 March
Ibodutant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Lanepitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
L-733,060
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Orvepitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Talnetant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Burapitant
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Vofopitant
InterPro Family
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Tachykinin_receptor
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Serlopitant
Chemical compound
may potentially make it useful in the treatment of asthma. Ibodutant Nepadutant Saredutant Beresford IJ, Sheldrick RL, Ball DI, Turpin MP, Walsh DM, Hawcock
GR-159897
Chemical compound
Vofopitant NK2 Agonists: Neurokinin A Antagonists: GR-159897 Ibodutant Nepadutant Saredutant Otilonium bromide NK3 Agonists: Neurokinin B Senktide Antagonists:
Befetupitant
NEPADUTANT
NEPADUTANT
NEPADUTANT
NEPADUTANT
Girl/Female
Hindu
Creation of God Shiva
Girl/Female
Arabic, Muslim
Protector; Messenger
Girl/Female
Indian, Telugu
Victory on Mind; Mind Controlling
Girl/Female
Bengali, Gujarati, Hindu, Indian, Jain, Kannada, Malayalam, Marathi, Sanskrit, Sindhi, Telugu
Woman
Girl/Female
American, British, English, Latin
Golden
Boy/Male
Hindu, Indian, Punjabi, Sanskrit, Sikh
The Devotees
Boy/Male
French
Friend.
Girl/Female
Irish
Derived from the name Evelyn or Evelina.
Girl/Female
Tamil
Revered
Boy/Male
Hindu, Indian, Marathi, Sanskrit
A Friend of the Gods
NEPADUTANT
NEPADUTANT
NEPADUTANT
NEPADUTANT
NEPADUTANT