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DASATINIB

  • Dasatinib
  • Chemical compound

    Dasatinib, sold under the brand name Sprycel among others, is a targeted therapy medication used to treat certain cases of chronic myelogenous leukemia

    Dasatinib

    Dasatinib

    Dasatinib

  • Chronic myelogenous leukemia
  • Type of blood cancer

    to TK inhibitors, four novel agents were later developed. The first, dasatinib, blocks several further oncogenic proteins, in addition to more potent

    Chronic myelogenous leukemia

    Chronic myelogenous leukemia

    Chronic_myelogenous_leukemia

  • Bcr-Abl tyrosine-kinase inhibitor
  • Pharmaceutical drug class

    except for T315I. Dasatinib is also not a substrate of multidrug P-glycoprotein efflux pumps like imatinib. Because of this dasatinib may be active in

    Bcr-Abl tyrosine-kinase inhibitor

    Bcr-Abl_tyrosine-kinase_inhibitor

  • Beacon Pharmaceuticals
  • Pharmaceutical company of Bangladesh

    sofosbuvir, afatinib, axitinib, brigatinib, baricitinib, cabozantinib, dasatinib, neratinib, eltrombopag, ibrutinib, lenvatinib, palbociclib, regorafenib

    Beacon Pharmaceuticals

    Beacon_Pharmaceuticals

  • Senolytic
  • Type of molecule that may be able to induce death of senescent cells

    are repurposed anti-cancer molecules, such as the chemotherapeutic drug dasatinib and the experimental small molecule navitoclax. Soluble urokinase plasminogen

    Senolytic

    Senolytic

  • MD Anderson Cancer Center
  • Hospital in Houston, Texas, U.S.

    2006: FDA Approval of Dasatinib and Nilotinib for Resistant Leukemia MD Anderson researchers demonstrate the efficacy of dasatinib and nilotinib, leading

    MD Anderson Cancer Center

    MD Anderson Cancer Center

    MD_Anderson_Cancer_Center

  • Hagop Kantarjian
  • targeted therapies, including tyrosine kinase inhibitors such as imatinib, dasatinib, nilotinib, and bosutinib, which have increased 10-year survival rates

    Hagop Kantarjian

    Hagop_Kantarjian

  • Tyrosine kinase
  • Enzyme

    symptoms. Among currently available inhibitors to treat CML are imatinib, dasatinib, nilotinib, bosutinib and ponatinib. Gastrointestinal stromal tumors (GIST)

    Tyrosine kinase

    Tyrosine kinase

    Tyrosine_kinase

  • Scleroderma
  • Group of autoimmune diseases resulting in abnormal growth of connective tissue

    alefacept, and the tyrosine kinase inhibitors, imatinib, nilotinib, and dasatinib. Experimental therapies under investigation include endothelin receptor

    Scleroderma

    Scleroderma

    Scleroderma

  • Proto-oncogene tyrosine-protein kinase Src
  • Mammalian protein found in humans

    kinases) have been developed for therapeutic use. One notable example is dasatinib which has been approved for the treatment of chronic myeloid leukemia

    Proto-oncogene tyrosine-protein kinase Src

    Proto-oncogene tyrosine-protein kinase Src

    Proto-oncogene_tyrosine-protein_kinase_Src

  • Philadelphia chromosome
  • Genetic abnormality in leukemia cancer cells

    features of the Abl kinase domain important for activity and inhibitor binding. A) first generation TKI imatinib, B) second generation TKI dasatinib

    Philadelphia chromosome

    Philadelphia chromosome

    Philadelphia_chromosome

  • Amitriptyline
  • Tricyclic antidepressant

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Amitriptyline

    Amitriptyline

    Amitriptyline

  • Tyrosine kinase inhibitor
  • Drug typically used in cancer treatment

    leukemia (CML) and later gefitinib and erlotinib aiming at the EGF receptor. Dasatinib is a Src tyrosine kinase inhibitor that is effective both as a senolytic

    Tyrosine kinase inhibitor

    Tyrosine kinase inhibitor

    Tyrosine_kinase_inhibitor

  • Protein kinase inhibitor
  • Enzymes that block actions of protein kinases

    functions to overcome other disease drivers. Kinase inhibitors such as dasatinib are often used in the treatment of cancer and inflammation. Some of the

    Protein kinase inhibitor

    Protein_kinase_inhibitor

  • Src inhibitor
  • agents. PP1, PP2 (kinase inhibitor) are both inhibitors of Lck and FynT. Dasatinib Rivera-Torres J, José ES (2019). "Src Tyrosine Kinase Inhibitors: New

    Src inhibitor

    Src inhibitor

    Src_inhibitor

  • Erythropoietin
  • Protein that stimulates red blood cell production

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Erythropoietin

    Erythropoietin

    Erythropoietin

  • Bafetinib
  • Chemical compound

    T315I) and some dasatinib resistant mutations. Bafetinib also has more affinity for Bcr-Abl than nilotinib (but less than dasatinib) but only targets

    Bafetinib

    Bafetinib

    Bafetinib

  • Vilazodone
  • Antidepressant medication

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Vilazodone

    Vilazodone

    Vilazodone

  • Insulin
  • Peptide hormone

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Insulin

    Insulin

    Insulin

  • Ciprofloxacin
  • Fluoroquinolone antibiotic

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Ciprofloxacin

    Ciprofloxacin

    Ciprofloxacin

  • List of antileukemic drugs
  • List of drugs given to treat leukemia

    Asparaginase Cladribine Clofarabine Cyclophosphamide Cytosine arabinoside Dasatinib Daunorubicin Decitabine Etoposide Fludarabine Gemtuzumab ozogamicin Idarubicin

    List of antileukemic drugs

    List_of_antileukemic_drugs

  • Acute lymphoblastic leukemia
  • Blood cancer characterized by overproduction of lymphoblasts

    Additionally, tyrosine kinase inhibitors (TKIs) such as imatinib and dasatinib are incorporated for Philadelphia chromosome-positive ALL, improving treatment

    Acute lymphoblastic leukemia

    Acute lymphoblastic leukemia

    Acute_lymphoblastic_leukemia

  • Nilotinib
  • Chemical compound

    lung-related adverse effects are rare when compared with imatinib and dasatinib, there is a case report of acute respiratory failure from diffuse alveolar

    Nilotinib

    Nilotinib

    Nilotinib

  • Imatinib
  • Chemical compound

    2008). "Target spectrum of the BCR-ABL inhibitors imatinib, nilotinib and dasatinib". Leukemia & Lymphoma. 49 (4): 615–619. doi:10.1080/10428190801896103

    Imatinib

    Imatinib

    Imatinib

  • Elranatamab
  • Medication

    Non-receptor bcr-abl Asciminib Bosutinib Dasatinib Imatinib Nilotinib Ponatinib Radotinib Src (Bosutinib Dasatinib) Janus kinase (JAK) Baricitinib Fedratinib

    Elranatamab

    Elranatamab

  • Quipazine
  • Chemical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Quipazine

    Quipazine

    Quipazine

  • Bristol Myers Squibb
  • American pharmaceutical company

    nivolumab acts by inducing the immune system to attack the tumor. Sprycel (dasatinib) Taxol (paclitaxel). At one time, BMS held the solitary contract to harvest

    Bristol Myers Squibb

    Bristol Myers Squibb

    Bristol_Myers_Squibb

  • Sildenafil
  • Drug for erectile dysfunction and hypertension

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Sildenafil

    Sildenafil

    Sildenafil

  • Brain-derived neurotrophic factor
  • Protein found in humans

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Brain-derived neurotrophic factor

    Brain-derived neurotrophic factor

    Brain-derived_neurotrophic_factor

  • Pyrimidinylpiperazine
  • Chemical compound

    pyrimidinylpiperazine derivatives are drugs, including: Buspirone – anxiolytic Dasatinib – anticancer agent Eptapirone – anxiolytic Gepirone – anxiolytic (indicated

    Pyrimidinylpiperazine

    Pyrimidinylpiperazine

    Pyrimidinylpiperazine

  • Cerebrolysin
  • Experimental drug for neurodegenerative disorders

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Cerebrolysin

    Cerebrolysin

  • Trastuzumab deruxtecan
  • Medication

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Trastuzumab deruxtecan

    Trastuzumab deruxtecan

    Trastuzumab_deruxtecan

  • D+Q
  • Topics referred to by the same term

    D+Q may refer to: Dasatinib#Dasatinib+Quercetin Drawn & Quarterly This disambiguation page lists articles associated with the title D+Q. If an internal

    D+Q

    D+Q

  • Dexamethasone
  • Corticosteroid medication

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Dexamethasone

    Dexamethasone

    Dexamethasone

  • Ponatinib
  • Medication

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Ponatinib

    Ponatinib

    Ponatinib

  • Alnespirone
  • Antidepressant and anxiolytic drug

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Alnespirone

    Alnespirone

    Alnespirone

  • Crystal Mackall
  • American physician and immunologist

    exhaustion can be reversed by transient T cell rest and demonstrated that dasatinib, a commonly prescribed oral drug, could be used to rest human T cells

    Crystal Mackall

    Crystal Mackall

    Crystal_Mackall

  • Asciminib
  • Chemical compound

    investigator-selected tyrosine kinase inhibitors (IS-TKIs) (imatinib, nilotinib, dasatinib, or bosutinib). The main efficacy outcome measure was major molecular

    Asciminib

    Asciminib

    Asciminib

  • Pulmonary hypertension
  • Increased blood pressure in lung arteries

    of exposure to drugs such as benfluorex (a fenfluramine derivative), dasatinib, cocaine, methamphetamine, ethanol leading to cirrhosis, and tobacco leading

    Pulmonary hypertension

    Pulmonary hypertension

    Pulmonary_hypertension

  • Insulin-like growth factor 1 receptor
  • Cell receptor protein found in humans

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Insulin-like growth factor 1 receptor

    Insulin-like growth factor 1 receptor

    Insulin-like_growth_factor_1_receptor

  • ATC code L01
  • Pharmaceutical drug classification

    Mitomycin L01DC04 Ixabepilone L01DC05 Utidelone L01EA01 Imatinib L01EA02 Dasatinib L01EA03 Nilotinib L01EA04 Bosutinib L01EA05 Ponatinib L01EA06 Asciminib

    ATC code L01

    ATC_code_L01

  • Testosterone
  • Primary male sex hormone

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Testosterone

    Testosterone

    Testosterone

  • Dehydroepiandrosterone
  • Chemical compound

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Dehydroepiandrosterone

    Dehydroepiandrosterone

    Dehydroepiandrosterone

  • Cobimetinib
  • Chemical compound

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Cobimetinib

    Cobimetinib

    Cobimetinib

  • Pulmonary arterial hypertension
  • High blood pressure in the pulmonary arteries

    due to drug or toxin exposures. Methamphetamines, the chemotherapeutic dasatinib and the appetite suppressant and diet drug fenfluramine are associated

    Pulmonary arterial hypertension

    Pulmonary arterial hypertension

    Pulmonary_arterial_hypertension

  • Insulin-like growth factor 1
  • Protein found in humans

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Insulin-like growth factor 1

    Insulin-like growth factor 1

    Insulin-like_growth_factor_1

  • WWTR1
  • Protein-coding gene in the species Homo sapiens

    extracellular matrix stiffness and tension using thiazovivin, cucurbitacin I, dasatinib, fluvastatin, and pazopanib, exhibited positive results in breast cancer

    WWTR1

    WWTR1

    WWTR1

  • ZINC000443438219
  • Pharmaceutical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    ZINC000443438219

    ZINC000443438219

    ZINC000443438219

  • Α-Ketoglutaric acid
  • Chemical compound

    Holland WL, Donato AJ, Lesniewski LA (February 2023). "Senolytic drugs, dasatinib and quercetin, attenuate adipose tissue inflammation, and ameliorate metabolic

    Α-Ketoglutaric acid

    Α-Ketoglutaric acid

    Α-Ketoglutaric_acid

  • Targeted therapy
  • Type of therapy

    replaced gefitinib in this setting. Sorafenib (Nexavar) Sunitinib (Sutent) Dasatinib (Sprycel) Lapatinib (Tykerb) Nilotinib (Tasigna) Bosutinib (Bosulif) Ponatinib

    Targeted therapy

    Targeted therapy

    Targeted_therapy

  • Vardenafil
  • Chemical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Vardenafil

    Vardenafil

    Vardenafil

  • Trimetazidine
  • Drug for angina pectoris sold under many brand names

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Trimetazidine

    Trimetazidine

    Trimetazidine

  • Regorafenib
  • Chemical compound

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Regorafenib

    Regorafenib

  • Piperazine
  • Chemical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Piperazine

    Piperazine

    Piperazine

  • Neurotrophic factors
  • Family of biomolecules

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Neurotrophic factors

    Neurotrophic_factors

  • Entrectinib
  • TKI inhibitor used for cancer treatment

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Entrectinib

    Entrectinib

    Entrectinib

  • Lorlatinib
  • Kinase inhibitor for treatment of non-small-cell lung cancer

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Lorlatinib

    Lorlatinib

    Lorlatinib

  • Itraconazole
  • Medication used to treat fungal infections

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Itraconazole

    Itraconazole

    Itraconazole

  • Ranolazine
  • Drug used to treat angina

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Ranolazine

    Ranolazine

    Ranolazine

  • Bevacizumab
  • Medication

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Bevacizumab

    Bevacizumab

  • Vascular endothelial growth factor
  • Protein involved in blood vessel growth

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Vascular endothelial growth factor

    Vascular_endothelial_growth_factor

  • PIPES
  • Chemical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    PIPES

    PIPES

    PIPES

  • Posaconazole
  • Pharmaceutical drug

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Posaconazole

    Posaconazole

    Posaconazole

  • KIT gene
  • Mammalian protein and protein-coding gene

    is not inhibited by imatinib. In those cases other inhibitors such as dasatinib Avapritinib or nilotinib can be used. Researchers investigated the dynamic

    KIT gene

    KIT gene

    KIT_gene

  • Trifluoromethylphenylpiperazine
  • Serotonergic drug

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Trifluoromethylphenylpiperazine

    Trifluoromethylphenylpiperazine

    Trifluoromethylphenylpiperazine

  • The Hallmarks of Cancer
  • 2000 paper by Hanahan and Weinberg

    Smith, S., Toban, N., Bazile, M., & Aloyz, R. (2013). Resistance to Dasatinib in primary chronic lymphocytic leukemia lymphocytes involves AMPK-mediated

    The Hallmarks of Cancer

    The Hallmarks of Cancer

    The_Hallmarks_of_Cancer

  • Infantile myofibromatosis
  • Rare tumor in infants originating in connective tissue

    but not the p.Asp850Val mutant. Two other tyrosine kinase inhibitors, dasatinib and ponatinib, do inhibit the p.Asp850Val mutant's tyrosine kinase activity

    Infantile myofibromatosis

    Infantile_myofibromatosis

  • Anti-VEGF
  • Medication which blocks growth of blood vessels

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Anti-VEGF

    Anti-VEGF

    Anti-VEGF

  • Nanjing Ange Pharmaceutical
  • Chinese pharmaceutical company

    Antineoplastic medicines, which include: Sunitinib Lapatinib Nilotinib Dasatinib Gefitinib Erlotinib Imatinib Canertinib It also produces relative pharmaceutical

    Nanjing Ange Pharmaceutical

    Nanjing_Ange_Pharmaceutical

  • Vemurafenib
  • Targeted cancer drug

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Vemurafenib

    Vemurafenib

    Vemurafenib

  • Enilospirone
  • Chemical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Enilospirone

    Enilospirone

    Enilospirone

  • Synthetic lethality
  • Cell death resulting from a deficiency of or interaction between in two or more genes

    of the DNA repair kinase ATR, or by exposure to the kinase inhibitor dasatinib. There are two pathways for homologous recombinational repair of double-strand

    Synthetic lethality

    Synthetic_lethality

  • ACD856
  • TrkA and TrkB positive modulator

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    ACD856

    ACD856

  • Meta-Chlorophenylpiperazine
  • Serotonergic drug

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Meta-Chlorophenylpiperazine

    Meta-Chlorophenylpiperazine

    Meta-Chlorophenylpiperazine

  • Testosterone (medication)
  • Medication and naturally occurring steroid hormone

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Testosterone (medication)

    Testosterone (medication)

    Testosterone_(medication)

  • Cyclizine
  • Medication for motion sickness or vertigo

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Cyclizine

    Cyclizine

    Cyclizine

  • List of antineoplastic agents
  • bradycardia, pneumonia, pneumonitis, kidney cyst, ARDS and liver failure. Dasatinib PO BCR-ABL, SRC family, c-Kit, EPHA2 and PDGFR-β kinase inhibitor. Philadelphia

    List of antineoplastic agents

    List_of_antineoplastic_agents

  • Trastuzumab
  • Medication

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Trastuzumab

    Trastuzumab

    Trastuzumab

  • Flibanserin
  • Medication

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Flibanserin

    Flibanserin

    Flibanserin

  • Lodenafil
  • Chemical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Lodenafil

    Lodenafil

    Lodenafil

  • Oncogenomics
  • Sub-field of genomics

    methyltransferase activity of EZH2, or with addition of the kinase inhibitor dasatinib. Another approach is to individually knock out each gene in a genome and

    Oncogenomics

    Oncogenomics

    Oncogenomics

  • Dehydroepiandrosterone sulfate
  • Chemical compound

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Dehydroepiandrosterone sulfate

    Dehydroepiandrosterone sulfate

    Dehydroepiandrosterone_sulfate

  • Dihexa
  • Chemical compound

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Dihexa

    Dihexa

    Dihexa

  • Mosunetuzumab
  • Monoclonal antibody

    Non-receptor bcr-abl Asciminib Bosutinib Dasatinib Imatinib Nilotinib Ponatinib Radotinib Src (Bosutinib Dasatinib) Janus kinase (JAK) Baricitinib Fedratinib

    Mosunetuzumab

    Mosunetuzumab

  • Timeline of aging research
  • gerontologists demonstrate a mechanism of anti-aging senolytics, in particular of Dasatinib plus Quercetin (D+Q) – an increase of α-Klotho as shown in mice, human

    Timeline of aging research

    Timeline_of_aging_research

  • Amivantamab
  • Monoclonal antibody

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Amivantamab

    Amivantamab

    Amivantamab

  • Cetuximab
  • Pharmaceutical drug

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Cetuximab

    Cetuximab

    Cetuximab

  • Encorafenib
  • Chemical compound

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Encorafenib

    Encorafenib

    Encorafenib

  • HER2
  • Mammalian protein found in humans

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    HER2

    HER2

    HER2

  • VCU-1012
  • Pharmaceutical compound

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    VCU-1012

    VCU-1012

    VCU-1012

  • Epidermal growth factor receptor
  • Transmembrane protein

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Epidermal growth factor receptor

    Epidermal growth factor receptor

    Epidermal_growth_factor_receptor

  • Clonal hypereosinophilia
  • Group of blood-based disorders

    transplantation (HSCT); a second patient wit this mutation failed treatment with dasatinib and also required HSCT. Patients bearing the V617F mutation exhibited

    Clonal hypereosinophilia

    Clonal_hypereosinophilia

  • Saracatinib
  • Chemical compound

    tyrosine kinase in cells displaying high level of lipid rafts. Bosutinib Dasatinib Hennequin LF, Allen J, Breed J, Curwen J, Fennell M, Green TP, et al.

    Saracatinib

    Saracatinib

    Saracatinib

  • Filgrastim
  • Medication

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Filgrastim

    Filgrastim

    Filgrastim

  • Accelerated phase chronic myelogenous leukemia
  • Medical condition

    fever, bone pain, and swollen spleen. Patients treated with imatinib, dasatinib, and nilotinib have shown meaningful rates of hematologic and cytogenetic

    Accelerated phase chronic myelogenous leukemia

    Accelerated_phase_chronic_myelogenous_leukemia

  • Radotinib
  • Chemical compound

    Administration (FDA) or the European Medicines Agency (EMA). Imatinib Nilotinib Dasatinib Bcr-Abl tyrosine-kinase inhibitors Kim SH, Menon H, Jootar S, Saikia T

    Radotinib

    Radotinib

    Radotinib

  • Nerve growth factor
  • Mammalian protein found in humans

    Agonists: Ancestim Stem cell factor Kinase inhibitors: Agerafenib Axitinib Dasatinib Imatinib Masitinib Nilotinib Pazopanib Quizartinib Sorafenib Sunitinib

    Nerve growth factor

    Nerve growth factor

    Nerve_growth_factor

  • Benzylpiperazine
  • Recreational drug

    Meclozine MT-45 Oxatomide SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone

    Benzylpiperazine

    Benzylpiperazine

    Benzylpiperazine

  • Engineered CAR T cell delivery
  • Delivery methods of CAR-T cells

    Hermann; Hudecek, Michael (Jul 2019). "The tyrosine kinase inhibitor dasatinib acts as a pharmacologic on/off switch for CAR T cells". Science Translational

    Engineered CAR T cell delivery

    Engineered_CAR_T_cell_delivery

  • Receptor tyrosine kinase
  • Class of enzymes

    PDGFR, Flt3 Renal cell carcinoma, GIST, Endocrine pancreatic cancer 2006 Dasatinib (Sprycel) Abl, Arg, KIT, PDGFR, Src Imatinib-resistant CML 2007 Nilotinib

    Receptor tyrosine kinase

    Receptor tyrosine kinase

    Receptor_tyrosine_kinase

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