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Medication used for major depressive disorder
Gepirone, sold under the brand name Exxua, is a medication used for the treatment of major depressive disorder. It is taken orally. Side effects of gepirone
Gepirone
Medication used to treat anxiety disorders
chain. Structural analogues of buspirone include other azapirones like gepirone, ipsapirone, perospirone, and tandospirone. A number of analogues are recorded
Buspirone
development pipeline include gepirone and FKB01MD for major depression, gepirone and FKW00GA for social anxiety disorder, gepirone for hypoactive sexual desire
Fabre-Kramer_Pharmaceuticals
Esketamine (Spravato) – non-competitive NMDA receptor antagonist, other actions Gepirone (Exxua) – 5-HT1A receptor partial agonist and α2-adrenergic receptor antagonist
List_of_antidepressants
Anxiolytic and antidepressant medication
of drugs and is closely related to other azapirones like buspirone and gepirone. Tandospirone was introduced for medical use in Japan in 1996 and in China
Tandospirone
Class of psychotropic drugs
21102-95-4 ) Buspirone (Buspar) Enilospirone (CERM-3,726) Eptapirone (F-11,440) Gepirone (Exxua) Ipsapirone (TVX-Q-7,821) MJ-7378 (CAS number: 21103-03-7 ) Revospirone
Azapirone
Protein family
at the α2A and α2B subtypes. 1-PP (active metabolite of buspirone and gepirone) Aripiprazole Asenapine Atipamezole Cirazoline Clozapine Efaroxan Fipamezole
Alpha-2_adrenergic_receptor
Serotonin receptor protein distributed in the cerebrum and raphe nucleus
efficacy in relieving anxiety and depression. Buspirone, tandospirone, and gepirone are currently approved for these indications in different parts of the
5-HT1A_receptor
Class of chemical compounds
Quipazine (2-piperazin-1-ylquinoline) Many azapirones such as buspirone, gepirone, and tandospirone produce 1-PP as a metabolite. Antianginals Ranolazine
Substituted_piperazine
Antidepressant medication
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Mirtazapine
Class of antidepressant medication
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Atypical_antidepressant
Species of psychoactive cactus
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Peyote
Drug for erectile dysfunction and hypertension
SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone Tandospirone Tirilazad
Sildenafil
Class of CNS depressant drugs
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Benzodiazepine
Gamma-aminobutyric acid analog
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Gabapentin
Pharmaceutical compound
other serotonin 5-HT1A receptor agonists, such as 8-OH-DPAT, buspirone, gepirone, F-15599 (NLX-101), and vilazodone, among others. On the other hand, the
TMU4142
List of pharmaceutical drugs under clinical development for treatment of depression
reuptake inhibitor Fluvoxamine (Luvox) – serotonin reuptake inhibitor Gepirone (Exxua) – serotonin 5-HT1A receptor partial agonist and α2-adrenergic receptor
List of investigational antidepressants
List_of_investigational_antidepressants
SSRI antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Escitalopram
Pharmaceutical drug classification
Pivagabine N06AX16 Venlafaxine N06AX17 Milnacipran N06AX18 Reboxetine N06AX19 Gepirone N06AX21 Duloxetine N06AX22 Agomelatine N06AX23 Desvenlafaxine N06AX24 Vilazodone
ATC_code_N06
Chemical compound
Buspirone – anxiolytic Dasatinib – anticancer agent Eptapirone – anxiolytic Gepirone – anxiolytic (indicated for Major depressive disorder) Ipsapirone – anxiolytic
Pyrimidinylpiperazine
Medication to prevent nausea and vomiting
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Ondansetron
Class of depressant drugs derived from barbituric acid
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Barbiturate
Muscle relaxant medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Cyclobenzaprine
Mushrooms containing psychoactive indole alkaloids
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Psilocybin_mushroom
SNRI medication
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Duloxetine
Protein-coding gene in the species Homo sapiens
Xylazine Atipamezole Idazoxan 1-PP (active metabolite of buspirone and gepirone) Asenapine BRL-44408 Clozapine Lurasidone Mianserin Mirtazapine Paliperidone
Alpha-2A_adrenergic_receptor
Class of antidepressant medication
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Selective serotonin reuptake inhibitor
Selective_serotonin_reuptake_inhibitor
Neurotransmission-modulating substance
appetite suppressants, and entactogens. Azapirones such as buspirone, gepirone, and tandospirone are 5-HT1A receptor partial agonists marketed primarily
Serotonin_receptor_agonist
Beta blocker medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Metoprolol
SNRI antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Desvenlafaxine
Type of medication
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Monoamine_oxidase_inhibitor
Benzodiazepine medication
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Lorazepam
Antihistamine drug
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Hydroxyzine
Experimental antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
B777-81
Tricyclic antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Amitriptyline
SNRI/SNDRI used to treat depression and other CNS pathologies (Alzheimer's)
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Flufenoxine
Beta blocker drug
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Propranolol
Stimulant and antidepressant drug
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Indriline
Medications that increase norepinephrine
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Norepinephrine reuptake inhibitor
Norepinephrine_reuptake_inhibitor
Minor cannabinoid
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Cannabigerol
Medication mainly used for depression and smoking cessation
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Bupropion
Typical antipsychotic medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Chlorpromazine
Weight loss medication
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Phentermine
Group of antidepressants
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Hydrazine_(antidepressant)
Pharmaceutical compound
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
N-Phosphonooxymethyl-DMT
DMT-infused smoking blend
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Changa_(drug)
5-HT2C receptor agonist
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
BMB-101
SSRI antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Fluvoxamine
Chemical element with atomic number 54 (Xe)
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Xenon
Colourless non-flammable greenhouse gas
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Nitrous_oxide
Pharmaceutical compound
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
IPALT
CHCl3, historical anaesthetic and common solvent
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Chloroform
Medication mainly used to treat gout
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Colchicine
South American psychoactive decoction
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Ayahuasca
Alpha-adrenergic agonist
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Clonidine
Irreversible non-selective MAO inhibitor and antidepressant drug
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Phenelzine
Atypical antipsychotic medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Olanzapine
Benzodiazepine sedative
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Diazepam
Chemical compound found in all domains of life with largely unexplored effects
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
S-Adenosyl_methionine
Chemical compound
several of the azapirones. Alnespirone Binospirone BMY-7,378 Buspirone Gepirone (Dimethyl variation) Mdl-72832 [113777-33-6] MDL73975 [159650-30-3] MJ-7378
Azaspirodecanedione
Pharmaceutical compound
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
EGX-B
Serotonin modulator antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Vortioxetine
Hormone and medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Adrenaline
Medication
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Flibanserin
Pharmaceutical compound
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
2,4,6-TMPEA-NBOMe
Antihypotensive medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Midodrine
Dopamine agonist medication
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Ropinirole
Antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Dazepinil
Atypical antipsychotic medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Quetiapine
SNRI antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Venlafaxine
Medications that relax muscles of the airways
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Beta-adrenergic_agonist
Class of chemical compounds
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Partial_lysergamide
Medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Tamsulosin
Long-acting bronchiodilator
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Formoterol
Pharmaceutical compound
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Dibutepinephrine
Class of medication used to treat depression and other conditions
5-HT1A receptor partial agonism • Other actions Buspirone (off-label) • Gepirone • Tandospirone 1980s Serotonin–norepinephrine reuptake inhibitors (SNRIs)
Antidepressant
Pharmaceutical compound
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
M.G._6669
Psychedelic drug
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Dimethyltryptamine
CNS depressant medication
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Phenibut
Medication for overactive bladder
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Mirabegron
Atypical antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Tianeptine
Drug class
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Serotonin 5-HT2A receptor antagonist
Serotonin_5-HT2A_receptor_antagonist
Gabapentinoid and Skeletal Muscle Relaxant
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Baclofen
Pharmaceutical compound
than certain other serotonin 5-HT1A receptor agonists like buspirone and gepirone. It shows favorable pharmacokinetics in rodents. The chemical synthesis
NLX-266
Entactogen, stimulant, and psychedelic drug of the amphetamine family
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
3,4-Methylenedioxyamphetamine
SSRI antidepressant
Agomelatine Amisulpride Dextromethorphan/bupropion Esketamine Etryptamine‡ Gepirone Indeloxazine Flupentixol Ketamine§ Medifoxamine‡ Metryptamine‡ Oxaflozane‡
Sertraline
Chemical compound
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
4-HO-MET
Muscle relaxant medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Tizanidine
Blood pressure medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Carvedilol
Psychedelic drug
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
2C-B
Drug for angina pectoris sold under many brand names
SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone Tandospirone Tirilazad
Trimetazidine
Psychedelic drug found in toads, mushrooms and plants
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Bufotenin
Fluoroquinolone antibiotic
SNC-80 Vanoxerine Pyrimidinylpiperazines Buspirone Dasatinib Eptapirone Gepirone Ipsapirone Piribedil Pyrimidinylpiperazine Revospirone Tandospirone Tirilazad
Ciprofloxacin
Atypical antipsychotic medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Clozapine
Antihistamine medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Cyproheptadine
Investigational generalized anxiety disorder drugs
September 2025. It is likely to become outdated with time. Gepirone (Ariza; BMY-13805; Exxua; Gepirone ER; MJ-13805; Org-33062; TGFK-07AD; TGFK07AD; Travivo;
List of investigational generalized anxiety disorder drugs
List_of_investigational_generalized_anxiety_disorder_drugs
Chemical compound
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Chloroethylclonidine
Benzodiazepine drug
e Anxiolytics (N05B) 5-HT1ARTooltip 5-HT1A receptor agonists Buspirone Gepirone Tandospirone GABAARTooltip GABAA receptor PAMsTooltip positive allosteric
Bromazepam
Group of chemical compounds
quetiapine, ziprasidone) Azapirones (e.g., buspirone, eptapirone (F-11440), gepirone, perospirone, tandospirone) Bay R 1531 Befiradol (NLX-112; F-13640) BMY-14802
Β-Carboline
Medication
paliperidone, quetiapine, risperidone, zotepine) Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone) BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine
Milsaperidone
GEPIRONE
GEPIRONE
GEPIRONE
GEPIRONE
Boy/Male
Hindu
Embellishment, To be charming
Girl/Female
Tamil
Truthful, Date
Male
English
Anglicized form of Hebrew Chammuw'el, HAMUEL means "heat of God." In the bible, this is the name of a man of Simeon. Also, according to pseudo-Dionysius, this is the name of an archangel.Â
Girl/Female
Australian, Finnish, Latin
Mild; Soft; Silky
Boy/Male
Indian
Lord of rivers, Ocean
Girl/Female
Italian Irish Latin
Lady. From the respectful title Donna.
Girl/Female
Arabic, Muslim
Moon of the Women
Boy/Male
Irish
Hero.
Boy/Male
Indian, Sanskrit
King of the Waters
Girl/Female
Indian, Punjabi, Sikh
Winning the Service of Guru's Lotus Feet
GEPIRONE
GEPIRONE
GEPIRONE
GEPIRONE
GEPIRONE