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DOTARIZINE

  • Dotarizine
  • Calcium channel blocker used in the treatment of migraine

    Dotarizine is a drug used in the treatment of migraine, which acts as a calcium channel blocker, and also as an antagonist at the 5-HT2A receptor, and

    Dotarizine

    Dotarizine

    Dotarizine

  • Migraine
  • Disorder resulting in recurrent moderate–severe headaches

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Migraine

    Migraine

  • Cyclobenzaprine
  • Muscle relaxant medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Cyclobenzaprine

    Cyclobenzaprine

    Cyclobenzaprine

  • Hydroxyzine
  • Antihistamine drug

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Hydroxyzine

    Hydroxyzine

    Hydroxyzine

  • Ibogaine
  • Psychoactive substance found in plants in the family Apocynaceae

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Ibogaine

    Ibogaine

    Ibogaine

  • Cocaine
  • Tropane alkaloid and stimulant drug

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Cocaine

    Cocaine

    Cocaine

  • Barbiturate
  • Class of depressant drugs derived from barbituric acid

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Barbiturate

    Barbiturate

    Barbiturate

  • Amlodipine
  • Medication against high blood pressure

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Amlodipine

    Amlodipine

    Amlodipine

  • Clonidine
  • Alpha-adrenergic agonist

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Clonidine

    Clonidine

    Clonidine

  • Β-Carboline
  • Group of chemical compounds

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Β-Carboline

    Β-Carboline

    Β-Carboline

  • Gabapentin
  • Gamma-aminobutyric acid analog

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Gabapentin

    Gabapentin

    Gabapentin

  • Dimethyltryptamine
  • Psychedelic drug

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Dimethyltryptamine

    Dimethyltryptamine

    Dimethyltryptamine

  • Ubrogepant
  • Medication for migraine headache acute treatment

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Ubrogepant

    Ubrogepant

    Ubrogepant

  • Atogepant
  • Chemical compound

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Atogepant

    Atogepant

    Atogepant

  • Ayahuasca
  • South American psychoactive decoction

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Ayahuasca

    Ayahuasca

    Ayahuasca

  • MDMA
  • Psychoactive drug, often called ecstasy

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    MDMA

    MDMA

    MDMA

  • LSD
  • Psychedelic drug

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    LSD

    LSD

    LSD

  • Ketamine
  • Dissociative anesthetic and anti-depressant

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Ketamine

    Ketamine

    Ketamine

  • Lorazepam
  • Benzodiazepine medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Lorazepam

    Lorazepam

    Lorazepam

  • Trazodone
  • Antidepressant medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Trazodone

    Trazodone

    Trazodone

  • Fluoxetine
  • SSRI antidepressant

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Fluoxetine

    Fluoxetine

    Fluoxetine

  • Mirtazapine
  • Antidepressant medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Mirtazapine

    Mirtazapine

    Mirtazapine

  • Rimegepant
  • Medication for acute migraine in adults

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Rimegepant

    Rimegepant

    Rimegepant

  • Aripiprazole
  • Atypical antipsychotic medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Aripiprazole

    Aripiprazole

    Aripiprazole

  • Lamotrigine
  • Anticonvulsant medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Lamotrigine

    Lamotrigine

    Lamotrigine

  • Amitriptyline
  • Tricyclic antidepressant

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Amitriptyline

    Amitriptyline

    Amitriptyline

  • Meclizine
  • Chemical compound

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Meclizine

    Meclizine

    Meclizine

  • Diphenhydramine
  • Antihistamine medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Diphenhydramine

    Diphenhydramine

    Diphenhydramine

  • Buprenorphine
  • Opioid used to treat pain and opioid use disorder

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Buprenorphine

    Buprenorphine

    Buprenorphine

  • Pregabalin
  • Anticonvulsant medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Pregabalin

    Pregabalin

    Pregabalin

  • Landipirdine
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Landipirdine

    Landipirdine

    Landipirdine

  • Ondansetron
  • Medication to prevent nausea and vomiting

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Ondansetron

    Ondansetron

    Ondansetron

  • Alcohol (drug)
  • Active ingredient in fermented drinks

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Alcohol (drug)

    Alcohol (drug)

    Alcohol_(drug)

  • Zavegepant
  • Medication for treatment of migraine

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Zavegepant

    Zavegepant

    Zavegepant

  • Peyote
  • Species of psychoactive cactus

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Peyote

    Peyote

    Peyote

  • Atomoxetine
  • Medication used to treat ADHD

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Atomoxetine

    Atomoxetine

    Atomoxetine

  • Olanzapine
  • Atypical antipsychotic medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Olanzapine

    Olanzapine

    Olanzapine

  • Sildenafil
  • Drug for erectile dysfunction and hypertension

    Clocinizine Cyclizine DBL-583 Diphenpipenol Diphenylmethylpiperazine Dotarizine DPI-221 DPI-287 DPI-3290 GBR-12,783 GBR-12,935 GBR-13,069 GBR-13,098 GBR-13

    Sildenafil

    Sildenafil

    Sildenafil

  • Psilocybin
  • Chemical compound found in some species of mushrooms

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Psilocybin

    Psilocybin

    Psilocybin

  • Tramadol
  • Synthetic opioid pain medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Tramadol

    Tramadol

    Tramadol

  • Centhaquine
  • Cardiovascular medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Centhaquine

    Centhaquine

    Centhaquine

  • 4-AcO-EPT
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    4-AcO-EPT

    4-AcO-EPT

    4-AcO-EPT

  • TMU4142
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    TMU4142

    TMU4142

  • 11-Chloroasimilobine
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    11-Chloroasimilobine

    11-Chloroasimilobine

    11-Chloroasimilobine

  • SB-224289
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    SB-224289

    SB-224289

    SB-224289

  • Guanfacine
  • Medication used for high blood pressure and ADHD

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Guanfacine

    Guanfacine

    Guanfacine

  • Morning glory
  • Common name for more than 1,000 species of flowering plants in the family Convolvulaceae

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Morning glory

    Morning glory

    Morning_glory

  • MW073
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    MW073

    MW073

    MW073

  • Fremanezumab
  • Pharmaceutical biological monoclonal antibody

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Fremanezumab

    Fremanezumab

  • Rizatriptan
  • Medication used for the treatment of migraine headaches

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Rizatriptan

    Rizatriptan

    Rizatriptan

  • Topiramate
  • Medication used to treat epilepsy and migraine

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Topiramate

    Topiramate

    Topiramate

  • Chlorpromazine
  • Typical antipsychotic medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Chlorpromazine

    Chlorpromazine

    Chlorpromazine

  • Quetiapine
  • Atypical antipsychotic medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Quetiapine

    Quetiapine

    Quetiapine

  • Risperidone
  • Antipsychotic medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Risperidone

    Risperidone

    Risperidone

  • Chloroform
  • CHCl3, historical anaesthetic and common solvent

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Chloroform

    Chloroform

  • Bromojimscaline
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Bromojimscaline

    Bromojimscaline

    Bromojimscaline

  • 2C2-NBOMe
  • Chemical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    2C2-NBOMe

    2C2-NBOMe

    2C2-NBOMe

  • Serotonin
  • Monoamine neurotransmitter

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Serotonin

    Serotonin

    Serotonin

  • Haloperidol
  • Typical antipsychotic medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Haloperidol

    Haloperidol

    Haloperidol

  • List of investigational headache and migraine drugs
  • Investigational antimigraine drugs

    serotonin 5-HT1B and 5-HT1D receptor agonist and triptan – migraine [81] Dotarizine (Dotaricin; FI-6026) – calcium channel blocker and serotonin 5-HT1A, 5-HT2A

    List of investigational headache and migraine drugs

    List_of_investigational_headache_and_migraine_drugs

  • Phentermine
  • Weight loss medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Phentermine

    Phentermine

    Phentermine

  • 5-Hydroxytryptophan
  • Chemical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    5-Hydroxytryptophan

    5-Hydroxytryptophan

    5-Hydroxytryptophan

  • Valerian (herb)
  • Species of flowering plant

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Valerian (herb)

    Valerian (herb)

    Valerian_(herb)

  • Benzonatate
  • Oral cough medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Benzonatate

    Benzonatate

  • Promethazine
  • Sedating antihistamine

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Promethazine

    Promethazine

    Promethazine

  • Naratriptan
  • Chemical compound

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Naratriptan

    Naratriptan

    Naratriptan

  • AOP-208
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    AOP-208

    AOP-208

  • Z5247692566
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Z5247692566

    Z5247692566

    Z5247692566

  • Trifluoroproscaline
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Trifluoroproscaline

    Trifluoroproscaline

    Trifluoroproscaline

  • Paliperidone palmitate
  • Atypical antipsychotic medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Paliperidone palmitate

    Paliperidone palmitate

    Paliperidone_palmitate

  • Carbamazepine
  • Anticonvulsant medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Carbamazepine

    Carbamazepine

    Carbamazepine

  • Isoergine
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Isoergine

    Isoergine

    Isoergine

  • O-Methylanhalonidine
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    O-Methylanhalonidine

    O-Methylanhalonidine

    O-Methylanhalonidine

  • Dextropropoxyphene
  • Withdrawn opioid medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Dextropropoxyphene

    Dextropropoxyphene

    Dextropropoxyphene

  • Suzetrigine
  • Non-opioid analgesic drug

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Suzetrigine

    Suzetrigine

    Suzetrigine

  • Nuciferine
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Nuciferine

    Nuciferine

    Nuciferine

  • Sumatriptan
  • Medication used for migraines & cluster headaches

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Sumatriptan

    Sumatriptan

    Sumatriptan

  • 4-HO-MET
  • Chemical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    4-HO-MET

    4-HO-MET

    4-HO-MET

  • Galcanezumab
  • Monoclonal antibody

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Galcanezumab

    Galcanezumab

    Galcanezumab

  • Α-Methyltryptophan
  • Serotonergic drug

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Α-Methyltryptophan

    Α-Methyltryptophan

    Α-Methyltryptophan

  • Verapamil
  • Calcium channel blocker medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Verapamil

    Verapamil

    Verapamil

  • Prucalopride
  • Drug used to treat chronic constipation

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Prucalopride

    Prucalopride

    Prucalopride

  • Vilazodone
  • Antidepressant medication

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Vilazodone

    Vilazodone

    Vilazodone

  • Cholesterol
  • Sterol biosynthesized by all animal cells

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Cholesterol

    Cholesterol

    Cholesterol

  • Erenumab
  • Chemical compound

    Sumatriptan Zolmitriptan Ditans Alniditan† Lasmiditan Others Dimetotiazine Dotarizine Iprazochrome Oxetorone Pizotifen CGRP-R antagonists Rimegepant Ubrogepant

    Erenumab

    Erenumab

    Erenumab

  • Colchicine
  • Medication mainly used to treat gout

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Colchicine

    Colchicine

    Colchicine

  • Substituted phenethylamine
  • Chemical class of organic compounds

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Substituted phenethylamine

    Substituted phenethylamine

    Substituted_phenethylamine

  • Piperazine
  • Chemical compound

    Clocinizine Cyclizine DBL-583 Diphenpipenol Diphenylmethylpiperazine Dotarizine DPI-221 DPI-287 DPI-3290 GBR-12,783 GBR-12,935 GBR-13,069 GBR-13,098 GBR-13

    Piperazine

    Piperazine

    Piperazine

  • Chlorphenamine
  • Antihistamine used to treat allergies

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Chlorphenamine

    Chlorphenamine

    Chlorphenamine

  • Borax combo
  • Designer drug combination mimicking MDMA

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Borax combo

    Borax combo

    Borax_combo

  • Mefenamic acid
  • Chemical compound

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Mefenamic acid

    Mefenamic acid

    Mefenamic_acid

  • Cannabigerol
  • Minor cannabinoid

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Cannabigerol

    Cannabigerol

    Cannabigerol

  • Thujone
  • Group of four possible stereoisomers found in various plants: a.o., absinthe and mint

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Thujone

    Thujone

    Thujone

  • Nefopam
  • Analgesic medication

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Nefopam

    Nefopam

    Nefopam

  • Lysergic acid propylamide
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Lysergic acid propylamide

    Lysergic acid propylamide

    Lysergic_acid_propylamide

  • 6-Hydroxytryptamine
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    6-Hydroxytryptamine

    6-Hydroxytryptamine

    6-Hydroxytryptamine

  • Para-Chlorophenethylamine
  • Chemical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Para-Chlorophenethylamine

    Para-Chlorophenethylamine

    Para-Chlorophenethylamine

  • Benzocaine
  • Local anaesthetic drug

    ω-Agatoxin TK ω-Conotoxin MVIIC Benidipine Bepridil Cilnidipine Cinnarizine Dotarizine Efonidipine Flunarizine Lamotrigine Levetiracetam Lomerizine Loperamide

    Benzocaine

    Benzocaine

    Benzocaine

  • 4-PrO-DiPT
  • Pharmaceutical compound

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    4-PrO-DiPT

    4-PrO-DiPT

    4-PrO-DiPT

  • Echinopsis pachanoi
  • Mescaline-containing cactus

    penbutolol, pindobind, pindolol, propranolol, tertatolol) BMY-7378 CSP-2503 Dotarizine Ergolines (e.g., metergoline) Flopropione GSK-958108 Lecozotan LY-206130

    Echinopsis pachanoi

    Echinopsis pachanoi

    Echinopsis_pachanoi

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